Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- Casein kinase II subunit alpha'
- Dual specificity mitogen-activated protein kinase kinase 3
- Dual specificity protein kinase CLK2
- Dual specificity protein kinase TTK
- Dual specificty protein kinase CLK1
- Haspin (465-798)
- Haspin (aa 465-798)
- MAP kinase ERK1
- MAP kinase ERK2
- Misshapen-like kinase 1 (MINK)
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 3
- Mitogen-activated protein kinase 9
- Mitogen-activated protein kinase kinase kinase kinase 4
- Serine/threonine-protein kinase 17A
- Serine/threonine-protein kinase Aurora-C
- Serine/threonine-protein kinase D1
- c-Jun N-terminal kinase 1 truncation (JNK1) (aa 1-363)
4 ΔG°
- SCH772984
- US8546404, 6
- Astrosclerin-3
- Beta-carbonic anhydrase
- Carbonate dehydratase
- Carbonic Anhydrase (hpCA)
- Carbonic Anhydrase IV
- Carbonic Anhydrase VA
- Carbonic Anhydrase VB
- Carbonic Anhydrase XIV
- Carbonic Anhydrase XV
- Carbonic anhydrase
- Carbonic anhydrase 1
- Carbonic anhydrase 12
- Carbonic anhydrase 2
- Carbonic anhydrase 4
- Carbonic anhydrase 6 (CA-VI)
- Carbonic anhydrase 7
- Carbonic anhydrase 9
- Carbonic anhydrase, alpha family
- Gamma-carbonic anhydrase
- 4-hydrazinylbenzene-1-sulfonamide
- CHEMBL7204
- aromatic/heteroaromatic sulfonamide 3
- hydrazide deriv. 14
- 25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrial
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome CYP26A1
- Cytochrome P450 11B1, mitochondrial
- Cytochrome P450 11B2 (CYP11B2)
- Cytochrome P450 17A1
- Cytochrome P450 24A1
- Cytochrome P450 26B1
- Cytochrome P450 2C19
- Cytochrome P450 2C8
- Cytochrome P450 2C9
- Cytochrome P450 3A
- Cytochrome P450 3A5
- Cytochrome P450 3A5 (CYP3A5)
- Multidrug resistance-associated protein 4
- P-glycoprotein 1 and 3 (MDR1a/MDR1b)
- Solute carrier family 22 member 1
- US8987315, Ketoconazole
- US9180183, Ketoconazole
- US9271963, Ketoconazole
- US9394290, KTZ (ketoconazole)
- US9963439, Ketoconazole
- Aurora B/Incenp
- Aurora kinase A/Targeting protein for Xklp2
- Cyclooxygenase-1 (COX-1)
- Dual specificity protein kinase TTK
- Heart phosphodiesterase
- Homo sapiens phosphodiesterase 2A (PDE2A)
- Phosphodiesterase (TcrPDEC)
- Phosphodiesterase 1
- Phosphodiesterase 3
- Phosphodiesterase 3 (PDE3)
- Phosphodiesterase 3A
- Phosphodiesterase 4
- Phosphodiesterase 4A
- Phosphodiesterase 5A
- Phosphodiesterase Type 3 (PDE3A)
- Phosphodiesterase Type 3 (PDE3B)
- cAMP-specific 3',5'-cyclic phosphodiesterase 4A
- cAMP-specific 3',5'-cyclic phosphodiesterase 4B
- cGMP-specific 3',5'-cyclic phosphodiesterase
- 6-methyl-2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridine-3-carbonitrile
- 6-methyl-2-oxo-5-pyridin-4-yl-1H-pyridine-3-carbonitrile
- CHEMBL189
- Milrinone
- Primacor
- US9242982, Milrinone
- US9249139, Milrinone
- GRIA1
- GRIA2
- GRIA3
- GRIK1
- Glutamate Carboxypeptidase II (GCPII)
- Glutamate receptor 1
- Glutamate receptor ionotropic AMPA
- Glutamate receptor ionotropic, AMPA 2
- Glutamate receptor ionotropic, AMPA 4
- Glutamate receptor ionotropic, kainate
- Glutamate receptor ionotropic, kainate 1
- Glutamate receptor ionotropic, kainate 2
- Grik5
- Ionotropic glutamate receptor kainate 2/5
- Metabotropic glutamate receptor 1
- Metabotropic glutamate receptor 2
- Metabotropic glutamate receptor 4 (mGluR4)
- Metabotropic glutamate receptor 6
- NMDA receptor subunit 2C (GluN2C)
- (2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl)propanoic acid
- 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid
- AMPA
- CHEMBL276815
- Aurora kinase A/Targeting protein for Xklp2
- Axin-1/Glycogen synthase kinase-3 beta
- Casein kinase I isoform alpha
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon
- LIM domain kinase 1
- Myosin light chain kinase, smooth muscle
- Myotonin-protein kinase
- PAK 1/CDC42
- Protein kinase N1
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase (P70S6K)
- Ribosomal protein S6 kinase alpha 1
- Serine/threonine-protein kinase MRCK-A
- Serine/threonine-protein kinase Sgk1
- Serine/threonine-protein kinase TBK1
- Tyrosine kinase non-receptor protein 2
- Tyrosine-protein kinase JAK2
27 IC50
- US9221808, 1bo
- US9221808, 1bo-HCl
- US9221808, 1bo-Mes
- 5-hydroxytryptamine receptor 1A
- Adrenergic Alpha
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Beta-3 adrenergic receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Multidrug and toxin extrusion protein 1
- Multidrug resistance-associated protein 4
- P-glycoprotein 1
- Potassium channel subfamily K member 10
- Potassium voltage-gated channel subfamily H member 2
- Solute carrier family 22 member 2
- Toll-like receptor 4
- Twik-RElated Potassium (K+) channel 1 (TREK1)
- Uridine-5'-diphosphoglucuronosyltransferase 1A1
- CHEMBL723
- Carvedilol
- Coreg
- Dilatrend
- Eucardic
- [3-(9H-carbazol-4-yloxy)-2-hydroxypropyl][2-(2-methoxyphenoxy)ethyl]amine
- Beta-chymotrypsin
- Beta-lactamase AmpC
- CDK2/Cyclin E/G1/S-specific cyclin E2
- CaM kinase II
- Cyclin-Dependent Kinase 4 (CDK4)
- Malate dehydrogenase
- Mixed Lineage Kinase 1 (MLK1)
- Mixed Lineage Kinase 3 (MLK3)
- Myosin light chain kinase, smooth muscle
- Protein Kinase C
- Protein kinase C (PKC)
- Protein kinase C alpha type
- Tyrosine-protein kinase JAK3
- Zinc finger protein GLI1
- Zinc finger protein GLI2
- cAMP-Dependent Protein Kinase (PKA)
- cAMP-dependent protein kinase (PKA)
- cAMP-dependent protein kinase catalytic subunit gamma
- cGMP-Dependent Protein Kinase
24 IC50
- 3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,22}]tricosa-1(16),2(10),4(9),5,7,11(15),17(22),18,20-nonaen-12-one
- CHEMBL16958
- K-252c
- α-Carbonic anhydrase (αCA)
- β-Carbonic anhydrase (βCA)
- Alpha carbonic anhydrase
- Alpha-carbonic anhydrase
- Astrosclerin-3
- Axin-1/Glycogen synthase kinase-3 beta
- Beta-carbonic anhydrase
- Carbonic Anhydrase VA
- Carbonic Anhydrase XIII
- Carbonic Anhydrase XV
- Carbonic anhydrase
- Carbonic anhydrase 1
- Carbonic anhydrase 2
- Carbonic anhydrase 4
- Carbonic anhydrase 6 (CA-VI)
- Carbonic anhydrase 7
- Carbonic anhydrase 9
- Carbonic anhydrase, alpha family
- Gamma-carbonic anhydrase
- CHEMBL19429
- CHEMBL69710
- CHLORIDE
- Cl-
- POTASSIUM CHLORIDE
- SODIUM CHLORIDE
- chloride
- chloride ion
- 5-hydroxytryptamine receptor 4 (5-HT4)
- Alkaline phosphatase placental-like
- Alkaline phosphatase, tissue-nonspecific isozyme
- Alpi
- Beta lactamase
- Collagenase 3
- Cyclooxygenase
- Gag-Pol polyprotein
- Genome polyprotein
- Intestinal alkaline phosphatase
- Lipoxygenase (LOX)
- Phospholipase A2
- Prostaglandin E synthase
- Prostaglandin G/H synthase (cyclooxygenase)
- TPA: Essential protein of the mitochondrial intermembrane space
- Toll-like receptor 9
- hypothetical protein SA1422
- perilipin-1
- perilipin-5
- (1E,6E)-1,7-bis(3-methoxy-4-oxidanyl-phenyl)hepta-1,6-diene-3,5-dione
- (1E,6E)-1,7-bis(4-hydroxy-3-methoxy-phenyl)hepta-1,6-diene-3,5-dione
- (1E,6E)-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,6-diene-3,5-dione
- CHEMBL140
- CURCUMIN
- Curcurmin
- Diferuloylmethane
- MLS000069631
- Natural yellow 3
- SMR000058237
- Turmeric yellow
- cid_969516
- Bfl-1
- Dual Specificity Protein Phosphatase 1
- Dual specificity phosphatase Cdc25B
- Glyceraldehyde-3-phosphate dehydrogenase liver
- Heat Shock 70kDa Protein 1
- Hematopoietic protein-tyrosine phosphatase (HEPTP)
- MKP-3
- POsterior Segregation family member (pos-1)
- Protein fosB
- Protein fosB/Transcription factor jun-D
- RecName: Full=Zinc finger protein mex-5
- Runt-Related Transcription Factor 1 Isoform AML1C
- Voltage-gated calcium channel subunit alpha Cav2.2
- cardiac alpha tropomyosin
- eukaryotic translation initiation factor 4 gamma, 1 isoform 4
- heat shock 70kDa protein 8 isoform 2
- large T antigen
- neuronal munc18-1 binding protein
- ubiquitin-conjugating enzyme E2 N
- 6-methoxy-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid
- MLS000072167
- SMR000009698
- cid_652912
- 5-hydroxytryptamine receptor 1A
- Cathepsin B
- Cathepsin S
- Dual Specificity Protein Phosphatase 1
- Dual specificity phosphatase Cdc25B
- Heat shock factor protein 1
- Heat shock protein HSP 90-alpha
- Heat shock protein HSP 90-beta
- Lipoamide Dehydrogenase (Lpd)
- MKP-3
- Nuclear receptor ROR-alpha
- Procathepsin L
- Pyruvate dehydrogenase (PDH)
- Serotonin (5-HT) receptor
- Sphingosine 1-phosphate receptor 1
- Sphingosine 1-phosphate receptor 3
- Steroidogenic Factor 1
- diphosphomevalonate decarboxylase
- mevalonate kinase
- 1-Ethyl-6-methyl-3-thiophen-2-yl-1H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione
- 1-ethyl-6-methyl-3-(2-thienyl)pyrimido[5,4-e][1,2,4]triazine-5,7-quinone
- 1-ethyl-6-methyl-3-thiophen-2-yl-pyrimido[5,4-e][1,2,4]triazine-5,7-dione
- 1-ethyl-6-methyl-3-thiophen-2-ylpyrimido[5,4-e][1,2,4]triazine-5,7-dione
- MLS000033110
- SMR000008918
- US9073941, 610
- cid_653297
- 5-hydroxytryptamine receptor 1A
- Angiotensin II receptor
- Apelin receptor
- Bcl-2-like protein 11
- DNA damage-inducible transcript 3 protein
- Histone acetyltransferase GCN5
- Histone acetyltransferase p300
- Inosine-5'-monophosphate dehydrogenase
- Inosine-5'-monophosphate dehydrogenase (IMPDH)
- Lanosterol synthase
- Nuclear receptor ROR-alpha
- Serotonin (5-HT) receptor
- Sphingosine 1-phosphate receptor 1
- Sphingosine 1-phosphate receptor 3
- Steroidogenic Factor 1
- Tumor necrosis factor
- XBP1
- nucleotide-binding oligomerization domain containing 1
- nucleotide-binding oligomerization domain containing 2
- 2-[(1,1-dioxido-1-benzothien-3-yl)thio]-5-phenyl-1,3,4-oxadiazole
- 3-[(5-phenyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-benzothiophene 1,1-dioxide
- 3-[(5-phenyl-1,3,4-oxadiazol-2-yl)thio]-1-benzothiophene 1,1-dioxide
- 3-[(5-phenyl-1,3,4-oxadiazol-2-yl)thio]benzothiophene 1,1-dioxide
- MLS000088644
- SMR000072650
- cid_890649
- Apoptosis regulator Bcl-2
- Axin-1/Glycogen synthase kinase-3 beta
- BCL-W
- Beta lactamase
- Bfl-1
- D(1A) dopamine receptor
- Dual Specificity Protein Phosphatase 1
- Ephrin type-B receptor 4
- Heat shock protein HSP 90-alpha
- Isoform Bcl-X(L)
- LANA
- MKP-3
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase kinase kinase kinase 2
- Serine/threonine-protein kinase 33
- Voltage-gated calcium channel subunit alpha Cav2.2
- beta-lactamase
- glutathione S-transferase
- metallo-beta-lactamase IMP-1
- MLS000080844
- SMR000044769
- cid_663844
- 3-hydroxy-3-methylglutaryl-coenzyme A reductase (HMG-CoA)
- Acetylcholinesterase
- Bfl-1
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cereblon/Histone deacetylase 6
- Cholinesterase
- Cystic fibrosis transmembrane conductance regulator
- HMG-CoA reductase
- Histone deacetylase 1
- Histone deacetylase 2
- Integrin alpha-L/beta-2 (LFA-1)
- Integrin beta-2/Leukocyte adhesion glycoprotein LFA-1 alpha
- Intercellular adhesion molecule (ICAM-1), Integrin alpha-L/beta-2
- Multidrug resistance-associated protein 4
- P-glycoprotein 1
- Solute carrier organic anion transporter family member 1B1 (OATP1B1)
- Sterol 14α-demethylase (CYP51)
- LOVASTATIN
- MLS000069585
- SMR000058779
- US9115116, lovastatin
- US9353061, Lovastatina
- cid_53232
- Apoptotic peptidase activating factor 1
- BZLF2
- Bfl-1
- Caspase-3
- Caspase-9
- Cathepsin B
- Dual Specificity Protein Phosphatase 1
- Dual specificity phosphatase Cdc25B
- Focal adhesion kinase 1
- MKP-3
- PPP5C protein
- PTK2B protein tyrosine kinase 2 beta (PTK2B)
- Phospholipase A2
- Procathepsin L
- SUMO-1-specific protease
- SUMO/sentrin specific peptidase family member 8
- cysteine protease ATG4B isoform a
- mothers against decapentaplegic homolog 3
- protein phosphatase 1, catalytic subunit, alpha isoform 3
29 IC50
- 3-anilino-2H-isoquinolin-1-one
- 3-anilinoisocarbostyril
- 3-anilinoisoquinolin-1(2H)-one
- 3-phenylazanyl-2H-isoquinolin-1-one
- MLS000043701
- SMR000020713
- cid_2142225
- Bromodomain adjacent to zinc finger domain protein 2A
- Bromodomain adjacent to zinc finger domain protein 2B
- Bromodomain and PHD finger-containing protein 3
- Bromodomain and WD repeat-containing protein 1
- Bromodomain testis-specific protein
- Bromodomain-containing protein 1
- Bromodomain-containing protein 2
- Bromodomain-containing protein 3
- Bromodomain-containing protein 4
- Bromodomain-containing protein 7
- CREB-binding protein
- Cat eye syndrome critical region protein 2
- E3 ubiquitin-protein ligase TRIM33
- Histone acetyltransferase KAT2A/KAT2B
- Probable global transcription activator SNF2L2
- Protein polybromo-1
- Transcription activator BRG1
- Transcription initiation factor TFIID subunit 1-like
- Transcription intermediary factor 1-alpha
- N-[3-(3-methyl-4-oxo-4,5,6,7-tetrahydro-2H-isoindol-1-yl)-4-phenoxyphenyl]methanesulfonamide
- US9776990, Example 40
- DNA dC->dU-editing enzyme APOBEC-3G
- G protein signalling regulator 19
- Gag-Pol polyprotein
- Induced myeloid leukemia cell differentiation protein Mcl-1
- MPI protein
- Mannose-6-phosphate isomerase
- RGS7
- Regulator of G-protein signaling 8
- diphosphomevalonate decarboxylase
- eukaryotic translation initiation factor 4 gamma, 1 isoform 4
- insulin-degrading enzyme isoform 1 precursor
- large T antigen
- mevalonate kinase
- phosphatase, orphan 1
- phosphomannomutase 2
- probable DNA dC->dU-editing enzyme APOBEC-3A
- regulator of G-protein signaling 4
- regulator of G-protein signalling 16
- streptokinase A precursor
- 2-(2-morpholin-4-yl-5-morpholin-4-ylsulfonyl-phenyl)-1,2-benzothiazol-3-one
- 2-(2-morpholin-4-yl-5-morpholin-4-ylsulfonylphenyl)-1,2-benzothiazol-3-one
- 2-(2-morpholino-5-morpholinosulfonyl-phenyl)-1,2-benzothiazol-3-one
- 2-[2-(4-morpholinyl)-5-(4-morpholinylsulfonyl)phenyl]-1,2-benzothiazol-3-one
- MLS000055722
- SMR000060745
- cid_2325815
- Alkaline phosphatase, tissue-nonspecific isozyme
- G protein signalling regulator 19
- Gag-Pol polyprotein
- M18 aspartyl aminopeptidase
- MPI protein
- Mannose-6-phosphate isomerase
- Procathepsin L
- RGS7
- Regulator of G-protein signaling 8
- diphosphomevalonate decarboxylase
- eukaryotic translation initiation factor 4 gamma, 1 isoform 4
- insulin-degrading enzyme isoform 1 precursor
- large T antigen
- mevalonate kinase
- neutrophil cytosolic factor 1
- phosphatase, orphan 1
- phosphomannomutase 2
- regulator of G-protein signaling 4
- regulator of G-protein signalling 16
- 2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-benzothiazol-3-one
- 2-(4-methyl-3-piperidin-1-ylsulfonylphenyl)-1,2-benzothiazol-3-one
- 2-(4-methyl-3-piperidinosulfonyl-phenyl)-1,2-benzothiazol-3-one
- 2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-one
- MLS000057572
- SMR000060796
- cid_2327953
- Apurinic-apyrimidinic endonuclease 1 (APE-1)
- Delta-type opioid receptor
- Dual specificity protein phosphatase (VHR)
- Heat shock protein HSP 90-beta
- Hematopoietic cell protein-tyrosine phosphatase 70Z-PEP
- Hematopoietic protein-tyrosine phosphatase (HEPTP)
- Lipoamide Dehydrogenase (Lpd)
- MPI protein
- Phospholipase A2
- Phospholipase C, gamma 1
- Phospholipase C-beta-3
- Pyruvate dehydrogenase (PDH)
- Ras-related C3 botulinum toxin substrate 1
- Trypanosoma brucei RNA editing ligase 1
- Tyrosine-protein kinase ABL1
- cell division cycle 42 (GTP binding protein, 25kDa)
- cysteine protease ATG4B isoform a
- exonuclease V (RecBCD complex), alpha chain
- tyrosyl-DNA phosphodiesterase 2
- 1,6-dimethyl-3-propyl-pyrimido[5,4-e][1,2,4]triazine-5,7-dione
- 1,6-dimethyl-3-propyl-pyrimido[5,4-e][1,2,4]triazine-5,7-quinone
- 1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dione
- MLS000718932
- SMR000291200
- US9073941, 617
- cid_3164059
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Cytochrome P450 2D6
- D(2) dopamine receptor
- D(3) dopamine receptor
- Monoamine transporter
- Norepinephrine transporter
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Transporter
- adrenergic Alpha2
- n-AChR
- (S,S)-reboxetine
- Reboxetine
- Vestra
- Cytochrome P450 1A
- Cytochrome P450 2B6
- Cytochrome P450 2C19
- Cytochrome P450 2C8
- Cytochrome P450 2C9
- Cytochrome P450 2D6
- Cytochrome P450 3A
- EFGR (L747-E749del, A750P)
- EGF-R Tyrosine Kinase Mutant (G719C)
- EGFR (G719S)
- EGFR (L861Q)
- EGFR E746-A750del
- EGFR L747-S752del, P753S
- EGFR L747-T750del
- EGFR S752-I759del
- Epidermal growth factor receptor
- Epidermal growth factor receptor(L858R)
- Epidermal growth factor receptor(L858R, T790M)
- Receptor tyrosine-protein kinase erbB-2
- US10246444, Example 40
- Bile salt export pump
- Cytochrome P450 3A
- N+/K+ ATPase alpha-4/beta-1
- Na,K-ATPase alpha1beta1
- Na,K-ATPase alpha2beta1
- Na,K-ATPase alpha2beta2
- Na,K-ATPase alpha2beta3
- Na,K-ATPase isoform alpha-1 (α1)
- Nuclear receptor ROR-gamma (RORC)
- P-glycoprotein (P-gp)
- P-glycoprotein 1
- P-glycoprotein 1 and 3 (MDR1a/MDR1b)
- Replicase polyprotein 1ab
- STAT3
- Sodium/potassium-transporting ATPase alpha-1 chain
- Solute carrier organic anion transporter family member 1A4
- Solute carrier organic anion transporter family member 1B1 (OATP1B1)
- Solute carrier organic anion transporter family member 1B3 (OATP1B3)
- Transcription Factor STAT1
- DIGOXIN
- MLS000069819
- SMR000059217
- US10668094, Compound Digoxin
- cid_2724385
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- Adrenergic alpha1B
- Alpha-1A adrenergic receptor
- Alpha-1D adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Histamine H1 receptor
- 3-(4-(3,6-dihydro-4-phenyl-1(2H)-pyridinyl)butyl)-1H-indol-5-ol
- 3-[4-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)butyl]-1H-indol-5-ol
- 3-[4-(4-phenyl-3,6-dihydropyridin-1(2H)-yl)butyl]-1H-indol-5-ol
- CHEMBL431367
- roxindole
- Bile salt export pump
- C-X-C chemokine receptor type 4 (CXCR4)
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- DNA polymerase beta
- HIV-1 B HXB2-LAI-IIIB-BRU
- HIV-1 protease
- Human immunodeficiency virus type 1 protease
- Human immunodeficiency virus type 1 reverse transcriptase
- Multidrug resistance-associated protein 4
- PKC alpha and beta-2
- Protein kinase C, epsilon
- Reverse Transcriptase
- Reverse transcriptase
- Serum albumin
- Thymidine kinase
- Thymidine kinase, cytosolic
- Thymidylate kinase
- Uridine-5'-diphosphoglucuronosyltransferase 2B7
- (AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
- (AZT)1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
- 1-((2R,4R,5S)-4-azido-5-(hydroxymethyl)tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione
- 1-((2R,4S,5S)-4-(diazoamino)-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione
- 1-((2R,4S,5S)-4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
- 1-((2R,4S,5S)-4-azido-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione
- 1-((2R,4S,5S)-4-azido-5-(hydroxymethyl)tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione
- 1-((2R,5S)-4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
- 1-((2S,4R,5R)-4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione (AZT)
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione (AzddThd, AZT)
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione (N3ddThd)
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione [AZT]
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione(3'-azido-2',3'-dideoxythymidine)
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione(AZT)
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione(Zidovudine, AZT)
- 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione(azidothymidine, AZT)
- 3'-Azido-3'-deoxy-thymidine
- 3'-Deoxy-3-azidothymidine
- 3'-azido-2',3'-dideoxythymidine
- 3'-azido-thymidine
- 3'azido-2'3'-dideoxythymidine
- 3-((2S,3S,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-3-yl)triaz-1-en-2-ium-1-ide
- 4-(4-Azido-5-hydroxy-tetrahydro-furan-2-yl)-5-methyl-3H-pyrazine-2,6-dione
- AZT
- BW-A-509U
- BWA509U
- CHEMBL129
- Retrovir
- US10071110, Compound AZT
- ZIDOVUDINE
- azidothymidine
- zidovudin
- zudovidine
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 6
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- D(2) dopamine receptor
- Dopamine receptor
- HTR6
- Metabotropic glutamate receptor 3
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- 8-[4-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-butyl]-8-aza-spiro[4.5]decane-7,9-dione
- CHEMBL1204189
- CHEMBL35057
- TIOSPERONE
- Acidic fibroblast growth factor
- Bone morphogenetic protein 2
- Bone morphogenetic protein 4
- Bone morphogenetic protein 6
- C-C motif chemokine 2
- C-C motif chemokine 5
- C-X-C motif chemokine 2
- Chemokine CXCL12
- Eotaxin
- Fibroblast growth factor 2
- Fibroblast growth factor 4
- Fibroblast growth factor 7
- Interferon gamma
- Platelet factor 4
- Proheparin-binding EGF-like growth factor
- Protein Wnt-3a
- Secreted frizzled-related protein 1
- Sonic hedgehog protein
- Vascular endothelial growth factor A
19 Kd
- CHEMBL3288260
- Acidic fibroblast growth factor
- Bone morphogenetic protein 2
- Bone morphogenetic protein 4
- Bone morphogenetic protein 6
- C-C motif chemokine 2
- C-C motif chemokine 5
- C-X-C motif chemokine 2
- Chemokine CXCL12
- Eotaxin
- Fibroblast growth factor 2
- Fibroblast growth factor 4
- Fibroblast growth factor 7
- Interferon gamma
- Platelet factor 4
- Proheparin-binding EGF-like growth factor
- Protein Wnt-3a
- Secreted frizzled-related protein 1
- Sonic hedgehog protein
- Vascular endothelial growth factor A
19 Kd
- CHEMBL3288258
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Alpha-1A adrenergic receptor
- Alpha-2C adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Histamine H1 receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Potassium voltage-gated channel subfamily H member 2
- Sodium-dependent serotonin transporter
- CHEMBL3290012
- Angiopoietin-1 receptor
- Epidermal growth factor receptor
- Ferrochelatase R115L (FECH)
- Fibroblast growth factor receptor 1
- Focal adhesion kinase 1/vascular endothelial growth factor receptor 3
- Hepatocyte growth factor receptor
- Insulin-like growth factor I receptor
- Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Platelet-derived growth factor receptor alpha
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RET kinase mutant (V804L)
- RET kinase mutant (V804M)
- Tyrosine-protein kinase receptor FLT3
- Tyrosine-protein kinase receptor UFO
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- BMS-907351
- CABOZANTINIB
- CHEBI:72317
- Cabometyx
- Cometriq
- US10183928, Cabozantinib
- US10202365, Compound Cabozantinib
- US10227329, Compound Cabozantinib
- US10273211, Compound Cabozantinib
- US10464902, Cabozantinib
- US10774070, Compound Cabozantinib
- XL-184
- cabozantinib s-malate
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- Adrenergic alpha1B
- Alpha-1A adrenergic receptor
- Alpha-1D adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Histamine H1 receptor
- (6,7-Dihydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dimethyl-ammonium
- TL99
- Acetylcholinesterase
- Adrenaline alpha1
- Adrenaline alpha2
- Choline Acetyltransferase
- Choline acetylase
- Choline transporter
- Creatine transporter
- Neuronal acetylcholine receptor
- Neuronal acetylcholine receptor Alpha-3/Beta-2
- Neuronal acetylcholine receptor Alpha-3/Beta-4
- Neuronal acetylcholine receptor protein alpha-2/beta-2 subunit
- Neuronal acetylcholine receptor protein alpha-4/beta-2 subunit
- Neuronal acetylcholine receptor protein alpha-4/beta-4 subunit
- Neuronal acetylcholine receptor subunit alpha-2
- Neuronal acetylcholine receptor subunit alpha-3
- Neuronal acetylcholine receptor subunit alpha-4
- Solute carrier family 22 member 1
- Solute carrier family 22 member 2
- n-AChR
- 2-hydroxy-N,N,N-trimethylethanaminium
- CHEMBL282468
- CHEMBL293410
- CHEMBL920
- N-trimethylethanolamine
- OXTRIPHYLLINE
- choline
- trimethylethanolamine
- 3C-like proteinase
- 3C-like proteinase (3CL-PRO)
- Beta amyloid A4 protein
- Bile salt export pump
- Cytochrome P450 1A
- Cytochrome P450 2C19
- Cytochrome P450 2C8
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 2J2
- Cytochrome P450 3A
- Heparanase
- Histamine N-methyltransferase
- Histidine-rich protein
- Phosphoehtnaolamine Methyltransferases 1 (PMT1)
- Phosphoehtnaolamine Methyltransferases 2 (PMT2)
- Phosphoethanolamine N-methyltransferase
- Potassium voltage-gated channel subfamily H member 2
- Replicase polyprotein 1ab
- 4-[(7-chloroquinolin-4-yl)amino]-2-[(diethylamino)methyl]phenol
- AMODIAQUINE
- CHEMBL682
- med.21724, Compound 188
- Adrenergic Alpha
- Bile salt export pump
- CHRM4
- Cytochrome P450 1A
- Cytochrome P450 2C19
- Cytochrome P450 2C8
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Histamine H1 receptor
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Potassium voltage-gated channel subfamily H member 2
- Solute carrier family 22 member 2
- CHEMBL900
- Dimethyl-[2-(phenyl-o-tolyl-methoxy)-ethyl]-amine
- Disipal
- Invagesic
- N,N-dimethyl-2-(phenyl(o-tolyl)methoxy)ethanamine
- Norflex
- Norgesic
- ORPHENADRINE
- Orphengesic
- CDK2/CycE
- CDK4/Cyclin D3
- CDK6/CycD3
- CDK7/Cyclin H/MNAT1
- Cyclin-Dependent Kinase 1 (CDK1)
- Cyclin-Dependent Kinase 2 (CDK2)
- Cyclin-Dependent Kinase 4 (CDK4)
- Cyclin-Dependent Kinase 5 (CDK5)
- Cyclin-Dependent Kinase 9 (CDK9)
- Cyclin-dependent kinase 1
- Dual specificity protein kinase CLK1/CLK4
- Dual specificity protein kinase CLK2
- Dual specificity protein kinase CLK3
- Epidermal growth factor receptor
- Interferon-induced, double-stranded RNA-activated protein kinase
- PKC alpha and beta-2
- Platelet-derived growth factor receptor
- Protein kinase C alpha type
- cAMP-dependent protein kinase (PKA)
- CHEMBL367625
- N*2*-((1R,2S)-2-Amino-cyclohexyl)-N*6*-(3-chloro-phenyl)-9-ethyl-9H-purine-2,6-diamine
- 17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3)
- Acid-sensing ion channel 1
- Aldo-keto reductase family 1 member C1
- Aldo-keto reductase family 1 member C2
- Aldo-keto reductase family 1 member C4 (AK1C4)
- Amiloride-sensitive cation channel 3
- Beta amyloid A4 protein
- Bile salt export pump
- COX-1
- Cyclooxygenase
- Cyclooxygenase-1 (COX-1)
- Cyclooxygenase-2 (COX-2)
- Fatty-acid amide hydrolase 1
- Intestinal fatty acid-binding protein (hIFABP)
- Liver fatty acid binding protein (rat L-FABP)
- Prostaglandin E synthase/G/H synthase 2
- Prostaglandin G/H synthase (cyclooxygenase)
- Serum albumin
- Solute carrier family 22 member 6
- (+-)-2-fluoro-alpha-methyl-4-biphenylacetic acid
- 2-(2-fluoro-[1,1'-biphenyl-4-yl])propanoic acid
- 2-(2-fluorobiphenyl-4-yl)propanoic acid
- 2-fluoro-alpha-methyl-(1,1'-biphenyl)-4-acetic acid
- 3-fluoro-4-phenylhydratropic acid
- Ansaid
- CHEMBL563
- FLURBIPROFEN
- US9630914, Compound A
- ALK tyrosine kinase receptor
- BDNF/NT-3 growth factors receptor
- Cytoplasmic tyrosine-protein kinase BMX
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Hepatocyte growth factor receptor
- High affinity nerve growth factor receptor
- Insulin receptor
- Macrophage colony-stimulating factor 1 receptor (CSF1R)
- Mast/stem cell growth factor receptor Kit
- NT-3 growth factor receptor
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase receptor FLT3
- Tyrosine-protein kinase receptor Tie-1
- Vascular endothelial growth factor receptor 2
19 IC50
- CHEMBL3582439
- 3-dehydroquinate synthase
- Alpha-(1,3)-fucosyltransferase VII
- Alpha-glucosidase MAL12
- Anthrax toxin receptor 2
- Carbonic Anhydrase XIV
- Carbonic anhydrase
- Carbonic anhydrase 1
- Carbonic anhydrase 12
- Carbonic anhydrase 2
- Carbonic anhydrase 4
- Carbonic anhydrase 6 (CA-VI)
- Carbonic anhydrase 7
- Carbonic anhydrase 9
- Dihydroorotate dehydrogenase (fumarate)
- M18 aspartyl aminopeptidase
- Procathepsin L
- Procollagen-proline,2-oxoglutarate-4-dioxygenase
- Tyrosinase
- Xanthine dehydrogenase
- 3,4-Dihydroxybenzoate, VIII
- 3,4-dihydroxybenzoic acid
- 4,5-Dihydroxybenzoic acid
- 4-Carboxy-1,2-dihydroxybenzene
- CHEMBL37537
- Protocatechuic acid
- Protocatechuic acid (M1)
- Protocatehuic acid
- cid_72
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Delta-type opioid receptor
- Histamine H1 receptor
- Kappa-type opioid receptor
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
19 Ki
- 1-(2-Methoxy-phenyl)-piperidine-4-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide
- CHEMBL195927
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 4 (5-HT4)
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Adrenergic alpha1B
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- 1-((S)-2-aminopropyl)-1H-indazol-6-ol
- CHEMBL371300
- Aldehyde oxidase
- Androgen receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome P450 2B1
- Cytochrome P450 2B6
- Cytochrome P450 3A
- Estradiol receptor beta (ERβ)
- Estrogen receptor
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Multidrug resistance-associated protein 4
- Nuclear receptor subfamily 1 group I member 3
- Solute carrier family 22 member 2
- Steroid 5-alpha-reductase
- Sulfotransferase 1A1 (SULT1A1)
- Testis-specific androgen-binding protein
- Uridine-5'-diphosphoglucuronosyltransferase 1A1
- 17-ethinyl-3,17-estradiol
- 17-ethinyl-3,17-oestradiol
- 17-ethinylestradiol
- 17alpha-Ethinyl estradiol
- 17alpha-ethynylestra-1,3,5(10)-triene-3,17beta-diol
- 17alpha-ethynylestradiol
- CHEMBL691
- ETHINYL ESTRADIOL
- Ethinylestradiol
- Ethynyl estradiol
- ethinyloestradiol
- Aurora kinase A/B
- Axin-1/Glycogen synthase kinase-3 beta
- Cyclin-dependent kinase 2
- Cytoplasmic tyrosine-protein kinase BMX
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon
- Interleukin-1 receptor-associated kinase 1
- Interleukin-1 receptor-associated kinase 4
- Non-receptor tyrosine-protein kinase TYK2
- Nuclear receptor subfamily 2 group C member 2
- Serine/threonine-protein kinase TBK1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase TXK
- Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
- Voltage-gated potassium channel
21 IC50
- CHEMBL4097255
- US10676460, Example 1
- 5-hydroxytryptamine receptor 2A
- Aldehyde oxidase
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- DRD1
- DRD2
- HTR4
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Multidrug resistance-associated protein 4
- Nuclear receptor subfamily 4 group A member 2/Retinoic acid receptor RXR-alpha
- Potassium voltage-gated channel subfamily H member 2
- Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Solute carrier family 22 member 2
- 1-(3-(4-(5-chloro-2-oxo-2,3-dihydrobenzo[d]imidazol-1-yl)piperidin-1-yl)propyl)-1H-benzo[d]imidazol-2(3H)-one
- 5-Chloro-1-{1-[3-(2-hydroxy-2,3-dihydro-benzoimidazol-1-yl)-propyl]-piperidin-4-yl}-2,3-dihydro-1H-benzoimidazol-2-ol
- 5-Chloro-1-{1-[3-(2-oxo-2,3-dihydro-benzoimidazol-1-yl)-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one(domperidone)
- 5-chloro-1-(1-(3-(2-oxo-2,3-dihydrobenzo[d]imidazol-1-yl)propyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
- 5-chloro-1-{1-[3-(2-oxo-2,3-dihydro-benzoimidazol-1-yl)-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one
- 6-Chloro-1-{1-[3-(2-oxo-2,3-dihydro-benzoimidazol-1-yl)-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one(Domperidone)
- CHEMBL219916
- DOMPERIDONE
- DOMPERIDONE5-Chloro-1-{1-[3-(2-oxo-2,3-dihydro-benzoimidazol-1-yl)-propyl]-piperidin-4-yl}-1,3-dihydro-benzoimidazol-2-one
- US9132134, Domperidone
- Acetylcholinesterase
- Amine oxidase (flavin-containing) A
- Amine oxidase [flavin-containing] B
- Apoptotic peptidase activating factor 1
- Caspase-9
- Chain E, Fragment Double-D From Human Fibrin
- Cruzipain
- Dihydrolipoamide dehydrogenase
- Dihydrolipoyl dehydrogenase
- Glutathione reductase
- Glutathione reductase (GR)
- Microtubule-associated protein Tau isoform 2N4R (Tau 2N4R)
- Microtubule-associated protein tau
- POsterior Segregation family member (pos-1)
- RecName: Full=Zinc finger protein mex-5
- Tau
- Thioredoxin reductase 1 (TrxR)
- lens epithelium-derived growth factor p75
- neutrophil cytosolic factor 1
1 ΔG°
- 3,7-bis(dimethylamino)phenothiazin-5-ium chloride
- Basic Blue 9
- CHEMBL405110
- Methylenblau
- Methylene Blue anhydrous
- Methylene blue
- Methylene blue (10)
- SAMPL5, CBC-G10
- azul de metileno
- bleu de methylene
- cid_6099
- methylthioninium chloride
- 12-Lipoxygenase (12-LOX)
- Acetylcholinesterase
- Arachidonate 5-lipoxygenase
- Beta-secretase 1
- Cholinesterases; ACHE & BCHE
- Cyclooxygenase
- Cyclooxygenase-1 (COX-1)
- Hematopoietic cell protein-tyrosine phosphatase 70Z-PEP
- LANA
- Phosphotyrosine protein phosphatase
- Probable low molecular weight protein-tyrosine-phosphatase
- Prostaglandin G/H synthase (cyclooxygenase)
- Protein-tyrosine phosphatase 1B
- Sarcoplasmic/endoplasmic reticulum calcium ATP-ase
- Sarcoplasmic/endoplasmic reticulum calcium ATPase 1
- Tyrosinase
- Tyrosine-protein phosphatase non-receptor type 12 (PTP-PEST)
- cAMP-specific 3',5'-cyclic phosphodiesterase 4D
- streptokinase A precursor
- CHEMBL464006
- Morusin
- Morusin, 3
- TCMDC-124149
- cid_5281671
- α-glucosidase
- β-galactosidase
- Acidic alpha-glucosidase
- Alpha-glucosidase
- Alpha-mannosidase
- Apelin receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Ceramide glucosyltransferase
- Glycogen debranching enzyme
- Lactase-phlorizin hydrolase
- Lysosomal acid glucosylceramidase
- Lysosomal alpha-glucosidase
- Lysosomal alpha-mannosidase
- Maltase-glucoamylase
- Multidrug resistance-associated protein 4
- Sucrase-isomaltase
- alpha-Glucosidase (α-Glucosidase)
- (2R,3R,4R,5S)-1-(2-hydroxyethyl)-2-(hydroxymethyl)piperidine-3,4,5-triol
- (2R,3R,4R,5S)-1-ethoxy-2-(hydroxymethyl)piperidine-3,4,5-triol
- BAY-M-1099
- CHEMBL1561
- Glyset
- MIGLITOL
- N-Hydroxyethyl-1-deoxynojirimycin
- cid_441314
- Angiopoietin-1 receptor
- Aurora kinase A/Targeting protein for Xklp2
- Aurora kinase B
- Cyclin-dependent kinase 2
- Cyclin-dependent kinase 4
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Focal adhesion kinase 1
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- Mitogen-activated protein kinase kinase kinase 8
- Platelet-derived growth factor receptor beta
- Proto-oncogene tyrosine-protein kinase Src
- Receptor tyrosine-protein kinase erbB-2
- Serine/threonine-protein kinase PLK4
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
19 IC50
- 4-[1-(tert-Butoxymethyl)-1H-indol-3-yl]-3-(3,4,5-trimethoxyphenyl)-1,5-dihydro-2H-pyrrole-2-one
- CHEMBL488646
- Cathepsin G
- Coagulation factor X
- Coagulation factor XI
- Coagulation factor XII
- Complement C1s
- Granzyme B
- Hepatocyte growth factor activator/Serine protease hepsin/Suppressor of tumorigenicity 14 protein
- Kallikrein 1
- Kallikrein 14
- Kallikrein 2
- Kallikrein 5
- Kallikrein 6
- Kallikrein-12
- Kallikrein-13
- Plasma kallikrein
- Plasminogen
- Prothrombin
- Thrombin and coagulation factor VII
- Vitamin K-dependent protein C
- CHEMBL4094403
- Cathepsin G
- Coagulation factor X
- Coagulation factor XI
- Coagulation factor XII
- Complement C1s
- Granzyme B
- Hepatocyte growth factor activator/Serine protease hepsin/Suppressor of tumorigenicity 14 protein
- Kallikrein 1
- Kallikrein 14
- Kallikrein 2
- Kallikrein 5
- Kallikrein 6
- Kallikrein-12
- Kallikrein-13
- Plasma kallikrein
- Plasminogen
- Prothrombin
- Thrombin and coagulation factor VII
- Vitamin K-dependent protein C
- CHEMBL4059991
- Cathepsin G
- Coagulation factor X
- Coagulation factor XI
- Coagulation factor XII
- Complement C1s
- Granzyme B
- Hepatocyte growth factor activator/Serine protease hepsin/Suppressor of tumorigenicity 14 protein
- Kallikrein 1
- Kallikrein 14
- Kallikrein 2
- Kallikrein 5
- Kallikrein 6
- Kallikrein-12
- Kallikrein-13
- Plasma kallikrein
- Plasminogen
- Prothrombin
- Thrombin and coagulation factor VII
- Vitamin K-dependent protein C
22 Ki
- CHEMBL4070056
- Cyclin-dependent kinase 1
- Cyclin-dependent kinase 2
- Cyclin-dependent kinase 4
- Epidermal growth factor receptor
- Histidine-tagged Rb
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin receptor
- MAP kinase-activated protein kinase 2
- Mitogen-activated protein kinase kinase kinase 8
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Protein kinase C theta type
- Proto-oncogene tyrosine-protein kinase Src
- RAC-alpha serine/threonine-protein kinase
- Serine/threonine-protein kinase B-raf
- Signal transducer and activator of transcription 3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Vascular endothelial growth factor receptor 2
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
19 IC50
- 4-[(4-Furan-3-yl-3-hydroxy-benzylamino)-methylene]-6-iodo-4Hisoquinoline-1,3-dione
- CHEMBL504547
- AMPK subunit alpha-2
- Axin-1/Glycogen synthase kinase-3 beta
- Cyclin-dependent kinase 2
- Dual specificity mitogen-activated protein kinase kinase 1
- Dual specificity mitogen-activated protein kinase kinase 4
- Dual specificity mitogen-activated protein kinase kinase 6
- Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin receptor
- MAP kinase-activated protein kinase 2
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 12
- Mitogen-activated protein kinase 13 (MAPK13)
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 8
- Mitogen-activated protein kinase 9
- Protein kinase C theta type
- Ribosomal protein S6 kinase (P70S6K)
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
- 4-(4-(2-(cyclopentylamino)pyrimidin-4-yl)-1H-pyrazol-3-yl)cyclohexanol
- CHEMBL507249
- Cell division control protein 42 homolog
- Cytochrome P450 1A
- Cytochrome P450 2C19
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Focal adhesion kinase 1
- Mitogen-activated protein kinase kinase kinase 11
- Protein kinase C delta type
- Protein kinase C, epsilon
- Protein kinase N2
- Rho-associated protein kinase 2
- Serine/threonine-protein kinase MST4
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase pim-2
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase Lyn
- Vascular endothelial growth factor receptor 1
- cGMP-dependent protein kinase
19 IC50
- 3,4-Dimethoxy-N-[3-(1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamide
- CHEMBL604087
- Androgen Receptor
- Bile acid receptor
- Estradiol receptor beta (ERβ)
- Estrogen receptor
- Glucocorticoid receptor
- Mineralocorticoid receptor
- Nuclear receptor subfamily 1 group I member 2
- Nuclear receptor subfamily 1 group I member 3
- Oxysterols receptor LXR-alpha
- Oxysterols receptor LXR-beta
- Peroxisome proliferator-activated receptor
- Peroxisome proliferator-activated receptor alpha (PPAR alpha)
- Peroxisome proliferator-activated receptor delta
- Progesterone receptor
- Retinoic acid receptor RXR-alpha
- Retinoid X receptor gamma/retinoic acid receptor alpha
- Retinoid receptor
- Thyroid hormone receptor alpha
- Vitamin D3 receptor
22 EC50
- 4-(((6-((3-(2,6-dichlorophenyl)-5-isopropylisoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
- CHEMBL1209109
- Androgen Receptor
- Bile acid receptor
- Estradiol receptor beta (ERβ)
- Estrogen receptor
- Glucocorticoid receptor
- Mineralocorticoid receptor
- Nuclear receptor subfamily 1 group I member 2
- Nuclear receptor subfamily 1 group I member 3
- Oxysterols receptor LXR-alpha
- Oxysterols receptor LXR-beta
- Peroxisome proliferator-activated receptor
- Peroxisome proliferator-activated receptor alpha (PPAR alpha)
- Peroxisome proliferator-activated receptor delta
- Progesterone receptor
- Retinoic acid receptor RXR-alpha
- Retinoid X receptor gamma/retinoic acid receptor alpha
- Retinoid receptor
- Thyroid hormone receptor alpha
- Vitamin D3 receptor
22 EC50
- 3-(((6-((5-cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
- CHEMBL1209170
- Androgen Receptor
- Bile acid receptor
- Estradiol receptor beta (ERβ)
- Estrogen receptor
- Glucocorticoid receptor
- Mineralocorticoid receptor
- Nuclear receptor subfamily 1 group I member 2
- Nuclear receptor subfamily 1 group I member 3
- Oxysterols receptor LXR-alpha
- Oxysterols receptor LXR-beta
- Peroxisome proliferator-activated receptor
- Peroxisome proliferator-activated receptor alpha (PPAR alpha)
- Peroxisome proliferator-activated receptor delta
- Progesterone receptor
- Retinoic acid receptor RXR-alpha
- Retinoid X receptor gamma/retinoic acid receptor alpha
- Retinoid receptor
- Thyroid hormone receptor alpha
- Vitamin D3 receptor
22 EC50
- 4-(((6-((5-cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
- CHEMBL1209173
- Adenosine Receptors A2a (A2a)
- Adenosine receptor A1
- Adenosine receptor A2a
- Adenosine receptor A3
- Calcium channel
- Calcium channel (Type L)
- Cav1.3/Cav beta3/Cav alpha2delta complex
- Cytochrome P450 3A
- Glutathione reductase (GR)
- Indoleamine 2,3-dioxygenase 1
- Indoleamine 2,3-dioxygenase 2
- P-glycoprotein 1
- Potassium voltage-gated channel subfamily H member 2
- Sodium channel protein type 7 subunit alpha
- Thromboxane-A synthase
- Transient receptor potential cation channel subfamily A member 1
- Voltage-gated L-type calcium channel
- Voltage-gated L-type calcium channel alpha-1C subunit
- Voltage-gated calcium channel
- (nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester
- 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester
- Adalat
- Adalat CC
- Afeditab cr
- BAY-A-1040
- NIFEDIPINE
- Nefidipine
- Procardia
- Procardia XL
- dimethyl 2,6-dimethyl-4-(2-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate
- ALK tyrosine kinase receptor
- Axin-1/Glycogen synthase kinase-3 beta
- CDK2/Cyclin E/G1/S-specific cyclin E2
- Cyclin B/Cyclin-Dependent Kinase 1 (CDK1)/G2/mitotic-specific cyclin B2/G2/mitotic-specific cyclin B3
- Dual specificity mitogen-activated protein kinase kinase 1
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 3
- Focal adhesion kinase 1
- Hepatocyte growth factor receptor
- Insulin-like growth factor I receptor
- Macrophage-stimulating protein receptor
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 8
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Proto-oncogene tyrosine-protein kinase Src
- RAF proto-oncogene serine/threonine-protein kinase
- Serine/threonine-protein kinase PLK1
- Vascular endothelial growth factor receptor 2
20 IC50
- CHEMBL1684800
- N-(5-Amino-1-(4-methoxybenzyl)-1H-pyrazol-4-yl)-5-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido)-2-methylbenzamide
- 3-phosphoinositide dependent protein kinase-1
- Apoptosis Signal-regulating Kinase 1 (ASK1)
- Aurora kinase A/Targeting protein for Xklp2
- Aurora kinase B
- Cyclin-dependent kinase 2
- Inhibitor of nuclear factor kappa-B kinase subunit alpha
- Insulin receptor
- Insulin-like growth factor I receptor
- Mitogen-activated protein kinase 8
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 1
- Ribosomal protein S6 kinase (P70S6K)
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase Sgk1
- TGF-beta receptor type-1
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase SYK
- Vascular endothelial growth factor receptor 2
22 IC50
- 6-(2-Amino-4-pyrimidinyl)-1H-indazol-3-amine
- 6-(2-aminopyrimidin-4-yl)-1H-indazol-3-amine
- CHEMBL1688215
- CDK2/CycE
- CDK6/cyclin D1
- CaM-kinase kinase beta
- Casein kinase I isoform alpha
- Cyclin-Dependent Kinase 1 (CDK1)
- Cyclin-Dependent Kinase 4 (CDK4)
- Cyclin-Dependent Kinase 7 (CDK7)
- Cyclin-Dependent Kinase 9 (CDK9)
- Cyclin-dependent kinase 2
- Cyclin-dependent kinase 4
- Cyclin-dependent kinase 6
- Cyclin-dependent kinase 7
- Cyclin-dependent kinase 8
- Cyclin-dependent-like kinase 5
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Insulin receptor-related protein
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 15
- Mitogen-activated protein kinase 3
19 IC50
- CHEMBL1234833
- CaM kinase IV
- Casein kinase I isoform delta
- Cyclin-dependent kinase 2
- Epidermal growth factor receptor
- Hepatocyte growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Interleukin-1 receptor-associated kinase 4
- Mitogen-activated protein kinase 1
- Protein kinase C alpha type
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase alpha-3
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase PLK3
- Testis-specific serine/threonine-protein kinase 2
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase Lck
- Vascular endothelial growth factor receptor 2
19 IC50
- CHEMBL1270795
- CDK2/CycE
- CDK3/E
- CDK7/Cyclin H/MNAT1
- Cyclin-Dependent Kinase 1 (CDK1)
- Cyclin-Dependent Kinase 2 (CDK2)
- Cyclin-Dependent Kinase 5 (CDK5)
- Cyclin-K
- Cyclin-dependent kinase 1
- Cyclin-dependent kinase 2
- Cyclin-dependent kinase 6
- Cyclin-dependent kinase 9
- Cyclin-dependent-like kinase 5
- Cytochrome P450 1A
- Cytochrome P450 2C19
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase receptor FLT3
25 IC50
- CHEMBL1944698
- 72 kDa type IV collagenase
- Collagenase 3
- Disintegrin and metalloproteinase domain-containing protein 17
- Interstitial collagenase
- Matrix metalloproteinase 10
- Matrix metalloproteinase 15
- Matrix metalloproteinase 16
- Matrix metalloproteinase 26
- Matrix metalloproteinase-12 (MMP12)
- Matrix metalloproteinase-14 (MMP14)
- Matrix metalloproteinase-20
- Matrix metalloproteinase-24
- Matrix metalloproteinase-25
- Matrix metalloproteinase-7 (MMP7)
- Matrix metalloproteinase-9
- Neutrophil collagenase
- Sodium-dependent noradrenaline transporter
- Stromelysin-1
- UDP-3-O-acyl-GlcNAc deacetylase (LpxC)
- CHEMBL1956115
- BDNF/NT-3 growth factors receptor
- Cytoplasmic tyrosine-protein kinase BMX
- High affinity nerve growth factor receptor
- Insulin receptor
- Insulin-like growth factor 1 receptor
- JNK1/JNK2
- Macrophage colony-stimulating factor 1 receptor (c-Fms)
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Neuronal proto-oncogene tyrosine-protein kinase Src
- Platelet-derived growth factor receptor beta
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Receptor-type tyrosine-protein kinase FLT3
- TPR/MET fusion protein
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor Tie-1
- Vascular endothelial growth factor receptor 1
19 IC50
- CHEMBL2037211
- Aurora kinase A/Targeting protein for Xklp2
- Epidermal growth factor receptor
- Hepatocyte growth factor receptor
- Insulin-like growth factor I receptor
- Macrophage colony-stimulating factor 1 receptor (CSF1R)
- Mast/stem cell growth factor receptor Kit
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAF proto-oncogene serine/threonine-protein kinase
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase pim-1
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
19 IC50
- CHEMBL2046883
- ALK tyrosine kinase receptor
- Fibroblast growth factor receptor 1
- Focal adhesion kinase 1
- High affinity nerve growth factor receptor
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase kinase kinase 9 (MLK1)
- Phosphorylase kinase
- Potassium voltage-gated channel subfamily H member 2
- Proto-oncogene tyrosine-protein kinase Src
- Serine/threonine-protein kinase SIK1
- Serine/threonine-protein kinase WNK3
- Testis-specific serine/threonine-protein kinase 2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 3
20 IC50
- CHEMBL2151321
- US8486966, 1
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 7
- Adrenergic receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Histamine H1 receptor
- Histamine H2 receptor
- Histamine H3 receptor
- Kappa-type opioid receptor
- Monoamine transporter
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M2 and M4
- Muscarinic acetylcholine receptor M5
- Sigma non-opioid intracellular receptor 1
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
- CHEMBL2203406
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Cytochrome P450 1A
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Histamine H1 receptor
- Histamine H2 Receptor
- Serotonin (5-HT) receptor
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
- 1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine
- CHEMBL2204360
- Lu-AA21004
- Trintellix
- brintellix
- vortioxetine hydrobromide
- Dual specificity protein phosphatase (VHR)
- Dual specificity protein phosphatase 15
- Dual specificity protein phosphatase 23 (VHZ)
- Fas-associated protein-tyrosine phosphatase 1 (FAP1)
- Hematopoietic cell protein-tyrosine phosphatase 70Z-PEP
- Hematopoietic protein-tyrosine phosphatase (HEPTP)
- Leukocyte common antigen
- Low molecular weight phosphotyrosine protein phosphatase
- Protein-tyrosine phosphatase 1B
- Protein-tyrosine phosphatase 1C
- Protein-tyrosine phosphatase MEG2 (PTP-Meg2)
- Receptor-type tyrosine-protein phosphatase beta (PTPβ)
- Receptor-type tyrosine-protein phosphatase epsilon (PTPε)
- Receptor-type tyrosine-protein phosphatase gamma
- Receptor-type tyrosine-protein phosphatase mu (PTPμ)
- Tyrosine-protein phosphatase non-receptor type 11
- Tyrosine-protein phosphatase non-receptor type 12 (PTP-PEST)
- Tyrosine-protein phosphatase non-receptor type 2
- Tyrosine-protein phosphatase non-receptor type 3 (PTPH1)
- CHEMBL2396719
- Dual specificity protein phosphatase (VHR)
- Dual specificity protein phosphatase 15
- Dual specificity protein phosphatase 23 (VHZ)
- Fas-associated protein-tyrosine phosphatase 1 (FAP1)
- Hematopoietic cell protein-tyrosine phosphatase 70Z-PEP
- Hematopoietic protein-tyrosine phosphatase (HEPTP)
- Leukocyte common antigen
- Low molecular weight phosphotyrosine protein phosphatase
- Protein-tyrosine phosphatase 1B
- Protein-tyrosine phosphatase 1C
- Protein-tyrosine phosphatase MEG2 (PTP-Meg2)
- Receptor-type tyrosine-protein phosphatase beta (PTPβ)
- Receptor-type tyrosine-protein phosphatase epsilon (PTPε)
- Receptor-type tyrosine-protein phosphatase gamma
- Receptor-type tyrosine-protein phosphatase mu (PTPμ)
- Tyrosine-protein phosphatase non-receptor type 11
- Tyrosine-protein phosphatase non-receptor type 12 (PTP-PEST)
- Tyrosine-protein phosphatase non-receptor type 2
- Tyrosine-protein phosphatase non-receptor type 3 (PTPH1)
19 IC50
- CHEMBL2396718
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 7
- Adenosine receptor A1
- Adenosine receptor A2a
- Adenosine receptor A3
- Alpha-1A adrenergic receptor
- Alpha-1D adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2C adrenergic receptor
- Cannabinoid receptor 1
- Cannabinoid receptor 2
- D(2) dopamine receptor
- Histamine H1 receptor
- Histamine H2 Receptor
- Sigma non-opioid intracellular receptor 1
- Somatostatin receptor type 2
- Somatostatin receptor type 4
23 Ki
- CHEMBL3104093
- ALK tyrosine kinase receptor
- Aurora kinase A/Targeting protein for Xklp2
- Casein kinase II subunit alpha
- Casein kinase II subunit alpha'
- Fibroblast growth factor receptor 1
- High affinity nerve growth factor receptor
- LIM domain kinase 1
- Non-receptor tyrosine-protein kinase TYK2
- Protein kinase C (PKC)
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Serine/threonine-protein kinase SIK1
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
24 IC50
- CHEMBL3116050
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Delta-type opioid receptor
- Kappa-type opioid receptor
- Monoamine transporter
- Mu-type opioid receptor
- Serotonin (5-HT) receptor
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
19 Ki
- CHEMBL4278465
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Delta-type opioid receptor
- Histamine H2 receptor
- Kappa-type opioid receptor
- Monoamine transporter
- Mu-type opioid receptor
- Serotonin (5-HT) receptor
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
19 Ki
- CHEMBL1644980
- Aurora kinase A/B
- Axin-1/Glycogen synthase kinase-3 beta
- Epidermal growth factor receptor
- Inhibitor of NF-kappa-B kinase alpha/beta
- Leucine-rich repeat serine/threonine-protein kinase 2
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase kinase kinase 5
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
- Rho-associated protein kinase 1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
20 IC50
- CHEMBL4474208
- Angiotensin-converting enzyme 2
- Beta-lactamase OXA-23
- Beta-lactamase VIM-1
- Carbapenem-hydrolyzing beta-lactamase KPC
- Catalase
- Cathepsin G
- Chymase
- Chymotrypsinogen B2
- Dipeptidyl peptidase 8/9
- Dipeptidyl peptidase 9
- Dipeptidyl peptidase II and dipeptidyl peptidase IV (DPP2 and DPP4)
- Endothelin-converting enzyme 1
- Interstitial collagenase
- Leukocyte elastase
- Matrix metalloproteinase-9
- Plasminogen
- Prothrombin
- Trypsin
- Urokinase-type plasminogen activator/surface receptor
- CHEMBL4633785
- 5-HT1
- 5-hydroxytryptamine receptor 2C
- Adrenergic Alpha
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-2 adrenergic receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- DRD1
- Dopamine receptor
- GST-MALT lymphoma-associated translocation (MALT1)
- Histamine H1 receptor
- Muscarinic acetylcholine receptor M2
- NADPH oxidase 1
- Pleiotropic ABC efflux transporter of multiple drugs
- Prion protein
- Serum albumin
- Sodium channel protein type I I alpha subunit
- Trypanothione reductase
- N,N-dimethyl-3-(10-phenothiazinyl)-1-propanamine;hydrochloride
- N,N-dimethyl-3-phenothiazin-10-yl-propan-1-amine;hydrochloride
- N,N-dimethyl-3-phenothiazin-10-ylpropan-1-amine;hydrochloride
- PROMAZINE
- SR-01000000228-4
- US9504692, Promazine
- cid_5887
- dimethyl(3-phenothiazin-10-ylpropyl)amine;hydrochloride
- 3-phosphoinositide dependent protein kinase-1
- Beta-galactosidase
- C-C chemokine receptor type 6 (CCR6)
- Casein kinase I isoform alpha
- Caspase-3
- Cyclin B/Cyclin-Dependent Kinase 1 (CDK1)/G2/mitotic-specific cyclin B2/G2/mitotic-specific cyclin B3
- Cyclin-Dependent Kinase 1 (CDK1)
- Cyclin-Dependent Kinase 5 (CDK5)
- Cyclin-dependent kinase 1
- Cyclin-dependent-like kinase 5
- Dual specificty protein kinase CLK1
- Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A
- Dual-specificity tyrosine-phosphorylation regulated kinase 2
- Glycogen Synthase Kinase-3, beta
- Glycogen synthase kinase-3
- Interferon-induced, double-stranded RNA-activated protein kinase
- SUMO-1-specific protease
- SUMO/sentrin specific peptidase family member 8
- streptokinase A precursor
- (2 Z,3 E)-6-Bromoindirubin-3 -oxime
- (3E)-6-bromo-3-[3-(hydroxyamino)indol-2-ylidene]oxindole
- 6-bromo-3-[(2Z,3E)-3-(hydroxyimino)-2,3-dihydro-1H-indol-2-ylidene]-2,3-dihydro-1H-indol-2-one
- 6-bromoindirubin-3 -oxime
- 6BIO
- CHEMBL409450
- indirubin deriv. 7a
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- HTR1D
- HTR6
- Serotonin 1B/1D receptor
- Serotonin 1d (5-HT1d) receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin 2a (5-HT2a) receptor
- Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
- Serotonin 3a (5-HT3a)/3b (5-HT3b)/3c (5-HT3c)/3d (5-HT3d)/3e (5-HT3e) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- 4-(4-Methyl-piperazin-1-yl)-7-trifluoromethyl-pyrrolo[1,2-a]quinoxaline
- CAS_109028-10-6
- CGS 12066B
- CHEMBL27403
- NSC_123945
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- Alpha-1A adrenergic receptor
- Beta-2 adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- GALANIN
- GRIA3
- Gamma-aminobutyric acid receptor subunit alpha-1
- Glutamate receptor ionotropic, NMDA 1
- HTR6
- Histamine H1 receptor
- Histamine H2 receptor
- Muscarinic acetylcholine receptor M2
- Serotonin (5-HT) receptor
- Serotonin 1B/1D receptor
- adrenergic Alpha2
- n-AChR
20 Ki
- CAS_3055171
- NAD-299
- NSC_3055171