Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- C-C motif chemokine 2
- Cell division control protein 42 homolog
- Myotonin-protein kinase
- Potassium voltage-gated channel subfamily H member 2
- Protein kinase C, epsilon
- Protein kinase N2
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Rho-associated protein kinase 2 (ROCK II)
- Rho-associated protein kinase 2/Transforming protein RhoA
- Rho-kinase (ROCK II)
- Ribosomal protein S6 kinase alpha 5
- cAMP-Dependent Protein Kinase (PKA)
- cAMP-Dependent Protein Kinase (PKA) Mutant (E127D)
- cAMP-Dependent Protein Kinase (PKA) Mutant (L49I)
- cAMP-Dependent Protein Kinase (PKA) Mutant (L49I/Q181K/T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (L49I/T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (L49I/V123M/E127D/Q181K/T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (L49I/V123M/Q181K/T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (Q181K/T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (V123M)
- cAMP-Dependent Protein Kinase (PKA) Mutant (V123M/Q181K/T183A)
- cAMP-Dependent Protein Kinase (PKA) Mutant (V123M/T183A)
- (R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXANECARBOXAMIDE
- 4-[(1R)-1-aminoethyl]-N-(pyridin-4-yl)cyclohexane-1-carboxamide
- US10183931, Y-27632
- Y-27632
- Bile salt export pump
- Bile salt export pump (BSEP)
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- DNA-dependent protein kinase
- Multidrug resistance-associated protein 4
- Myosin light chain kinase, smooth muscle
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
- Phosphoinositide 3-Kinase (PI3K), delta
- Phosphoinositide 3-Kinase (PI3K), gamma
- Polo-Like Kinase 3
- Polo-Like Kinase 4
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase PLK2
- Serine/threonine-protein kinase PLK3
- endothelial PAS domain-containing protein 1
- mRNA interferase toxin, antitoxin is MazE
- mTOR/FKBP12A/FKBP12B
- p110α/p85α
- p110β/p85α
- (1R,3R,5S,9R,18S)-18-(methoxymethyl)-1,5-dimethyl-6,11,16-trioxo-13,17-dioxapentacyclo[10.6.1.0^{2,10}.0^{5,9}.0^{15,19}]nonadeca-2(10),12(19),14-trien-3-yl acetate
- CHEMBL428496
- NSC221019
- Wortmannin
- Wortmannin, Wm
- cid_312145
- Adrenergic Alpha
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome P450 2J2
- DHFR
- Dihydrofolate Reductase (DHFR)
- Dihydrofolate Reductase (DHFR) Mutant (F98Y)
- Dihydrofolate Reductase (DHFR) Mutant (I100L)
- Dihydrofolate Reductase-Thymidylate Synthase (DHFR-TS) Mutant KICB1
- Dihydrofolate reductase
- Dihydrofolate reductase (DHFR)
- Dihydrofolate reductase (DfrA)
- Dihydrofolate reductase (DfrG)
- Dihydrofolate reductase (DfrK)
- Dihydrofolate reductase type 1
- Dihydrofolate reductase; P. carinii vs rat
- Dihydrofolate reductase; T. gondii vs rat
- Multidrug resistance-associated protein 4
- NH(3)-dependent NAD(+) synthetase
- Potassium voltage-gated channel subfamily H member 2
- Solute carrier family 22 member 1
- Trace amine-associated receptor 5
- protein-arginine deiminase type-4
- 5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-diamine
- CHEMBL22
- TMP
- Trimethoprim
- Trimethoprim (TMP)
- US10870625, Compound TMP
- Acidic alpha-glucosidase
- Alpha glucosidase
- Alpha-glucosidase
- Alpha-mannosidase 2C1
- Beta-galactosidase
- Beta-glucosidase
- Beta-mannosidase
- Ceramide glucosyltransferase
- Glucocerebrosidase GBA1/GBA2
- Glycogen debranching enzyme
- Lactase-glycosylceramidase
- Lactase-phlorizin hydrolase
- Lysosomal acid glucosylceramidase
- Lysosomal alpha-glucosidase
- Maltase-glucoamylase
- Mannosidase 2 alpha 1
- Mannosidase 2, alpha B1
- Non-lysosomal glucosylceramidase
- Sucrase-isomaltase
- Trehalase
- Uncharacterized protein
- alpha-Glucosidase (α-Glucosidase)
- alpha-Glucosidase (alpha-Glu)
- alpha-glucosidase (Gaa)
- (2R,3R,4R,5S)-1-butyl-2-(hydroxymethyl)piperidine-3,4,5-triol
- CHEMBL1029
- MIGLUSTAT
- N-Butyl-DNJ
- US9181184, 5
- β-lactamase (Bla2)
- ACEI-ACE2
- Angiotensin-Converting Enzyme
- Angiotensin-converting enzyme
- Bacterial beta-lactamase TEM
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cyclooxygenase
- Endothelin-converting enzyme 1 (ECE1)
- Endothelin-converting enzyme 2 (ECE-2)
- Leukotriene A-4 hydrolase
- Leukotriene A4 hydrolase
- Metallo-beta-lactamase VIM-2 (VIM-2)
- Metallo-beta-lactamase type 2
- Multidrug resistance-associated protein 4
- Neprilysin
- Neutral Endopeptidase (NEP)
- Prostaglandin E synthase/G/H synthase 2
- Prothrombin
- Renin
- Solute carrier family 15 member 1
- Succinyl-diaminopimelate desuccinylase
- metallo-beta-lactamase IMP-1
- (2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolidine-2-carboxylic acid
- CHEMBL1560
- Capozide
- Captopril
- Lopirin
- SQ 14,225
- SQ14534
- 1,3-beta-glucan synthase component GLS2
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome P450 11A1
- Cytochrome P450 3A
- DNA Gyrase
- DNA Gyrase Subunit A
- DNA Topoisomerase IV
- DNA Topoisomerase IV Subunit A
- DNA gyrase
- DNA gyrase subunit A
- DNA gyrase subunit A/DNA gyrase subunit B
- DNA gyrase subunit B
- DNA topoisomerase II
- Histamine H3 receptor
- Human immunodeficiency virus type 1 integrase
- Multidrug resistance protein mdtK
- Multidrug resistance-associated protein 4
- Potassium voltage-gated channel subfamily H member 2
- Topoisomerase I/II
- Topoisomerase IV
- Topoisomerase IV subunit A
- UvrD helicase (PfUDN)
- 1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid
- 1-cyclopropyl-6-fluoro-4-oxo-7-piperazin-1-yl-1,4-dihydroquinoline-3-carboxylic acid
- Bay 09867
- CHEMBL8
- Ciprinol
- Cipro
- Ciprofloxacin
- US9138393, Ciprofloxacin HCl
- US9144538, Ciprofloxacin HCl
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Carbonic anhydrase 1
- Carbonic anhydrase 2
- Cyclooxygenase
- Cyclooxygenase-1 (COX-1)
- Cyclooxygenase-2 (COX-2)
- Epidermal growth factor receptor
- GTP-binding protein (rab7)
- Gamma-glutamyltranspeptidase 1
- Integrin alpha-IIb/beta-3
- Liver fatty acid binding protein (rat L-FABP)
- Multidrug resistance-associated protein 4
- Myeloperoxidase
- Prostaglandin E synthase/G/H synthase 2
- Prostaglandin G/H synthase (Cyclooxygenase-2)
- Prostaglandin G/H synthase (cyclooxygenase)
- Ras-related C3 botulinum toxin substrate 1
- Ras-related protein Rab-2A.
- Solute carrier family 22 member 20
- Solute carrier family 22 member 6
- cell division cycle 42 (GTP binding protein, 25kDa)
- ras protein
- 2-(acetyloxy)benzoate
- 2-(acetyloxy)benzoic acid
- Acetylsalicylic acid
- Aspirin
- Endosprin
- Polopirin
- Zorprin
- acetylsalicylate
- cid_2244
- Angiopoietin-1 receptor
- Aurora kinase B
- Axin-1/Glycogen synthase kinase-3 beta
- Discoidin domain-containing receptor 2
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 1
- Fibroblast growth factor receptor 2
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Glycogen Synthase Kinase 3 (GSK3)
- Insulin receptor
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Polo-Like Kinase 3
- Polo-Like Kinase 4
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase PLK2
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor A
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
- 3-[(4-bromo-2,6-difluorophenyl)methoxy]-5-({[4-(pyrrolidin-1-yl)butyl]carbamoyl}amino)-1,2-thiazole-4-carboxamide
- CHEMBL253969
- CP 547632
- CP547632, 24
- US9446026, 1
- β-Carbonic anhydrase 2 (CA 2)
- Alpha carbonic anhydrase
- Astrosclerin-3
- Carbonate dehydratase
- Carbonic Anhydrase (mtCA 1)
- Carbonic Anhydrase (mtCA 3)
- Carbonic Anhydrase 2 (Can2)
- Carbonic Anhydrase III
- Carbonic Anhydrase VA
- Carbonic Anhydrase VB
- Carbonic Anhydrase XIV
- Carbonic Anhydrase XV
- Carbonic anhydrase
- Carbonic anhydrase 1
- Carbonic anhydrase 12
- Carbonic anhydrase 13 (CA XIII)
- Carbonic anhydrase 2
- Carbonic anhydrase 4
- Carbonic anhydrase 6 (CA-VI)
- Carbonic anhydrase 7
- Carbonic anhydrase 9
- Carbonic anhydrase, alpha family
- Delta carbonic anhydrase
- beta-Carbonic Anhydrase
76 Ki
- 4-(1,1-dioxo-1,2-thiazinan-2-yl)benzene-1-sulfonamide
- CHEMBL328560
- Contravul
- Ospolot
- Sulthiame (SLT)
- Sulthiame, 2
- Apoptotic peptidase activating factor 1
- Apurinic-apyrimidinic endonuclease 1 (APE-1)
- Caspase-9
- DNA recombination protein RecA
- Heat shock protein HSP 90-beta
- Hematopoietic cell protein-tyrosine phosphatase 70Z-PEP
- Hematopoietic protein-tyrosine phosphatase (HEPTP)
- Lipoamide Dehydrogenase (Lpd)
- MPI protein
- MSRA protein
- Phospholipase A2
- Pyruvate dehydrogenase (PDH)
- Serine/threonine-protein kinase PLK1
- Sphingosine 1-phosphate receptor 2
- Trypanosoma brucei RNA editing ligase 1
- Tyrosine-protein kinase ABL1
- Valosin-containing protein
- cell division cycle 42 (GTP binding protein, 25kDa)
- cysteine protease ATG4B isoform a
- mothers against decapentaplegic homolog 3
- nuclear receptor corepressor 2 isoform 2
- photoreceptor-specific nuclear receptor
- streptokinase A precursor
- tyrosyl-DNA phosphodiesterase 2
- 1,3,6-Trimethyl-1H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione
- 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione
- 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-quinone
- MLS000528498
- SMR000121073
- US9073941, 611
- cid_460747
- Bile salt export pump
- Organic anion-transporting polypeptide 1D1 (Oatp1d1)
- PTGDR
- PTGER3
- PTGER4
- PTGFR
- PTGIR
- Prostaglandin D Synthase
- Prostaglandin E2 receptor
- Prostaglandin E2 receptor EP1 subtype (EP1)
- Prostaglandin E2 receptor EP2 subtype
- Prostaglandin E2 receptor EP4 subtype
- Prostaglandin F2-alpha receptor
- Prostaglandin Transporter
- Prostanoid EP1 Receptor
- Prostanoid EP2 Receptor
- Prostanoid EP2 receptor
- Prostanoid EP3 Receptor
- Prostanoid EP4 Receptor
- Prostanoid EP4 receptor
- Prostanoid IP receptor
- Solute carrier family 22 member 20
- Solute carrier family 22 member 6
- TBXA2R
- (15S)-prostaglandin E2
- (5Z,11alpha,13E,15S)-11,15-dihydroxy-9-oxoprosta-5,13-dien-1-oic acid
- (5Z,13E,15S)-11alpha,15-dihydroxy-9-oxoprosta-5,13-dien-1-oic acid
- (E,Z)-(1R,2R,3R)-7-(3-Hydroxy-2-((3S)-(3-hydroxy-1-octenyl))-5-oxocyclopentyl)-5-heptenoic acid
- CHEMBL548
- DINOPROSTONE
- PGE2
- [3H]Dinoprostone
- [3H]PGE2
- [3H]Prostaglandin E2
- prostaglandin E2
- Acyl-CoA: cholesterol acyltransferase (ACAT)
- Aldehyde reductase
- Aldehyde reductase (ALR1)
- Aldose reductase
- Aldose reductase (ALR2)
- Aldose reductase-related protein 1
- Bile salt export pump
- Bile salt export pump (BSEP)
- Carboxylesterase 2
- Cereblon/Histone deacetylase 1
- Cereblon/Histone deacetylase 6
- Coagulation factor VII/tissue factor
- Cytochrome P450 2A6
- Histone deacetylase
- Histone deacetylase 1
- Histone deacetylase 2
- Histone deacetylase 3
- Histone deacetylase 4
- Histone deacetylase 5
- Histone deacetylase 7
- Histone deacetylase 8
- Histone deacetylase 9
- NAD-dependent protein deacetylase sirtuin-5 (SIRT5)
- Uridine-5'-diphosphoglucuronosyltransferase 2B7
- 2-n-propyl-n-valeric acid
- CHEMBL109
- DPA
- Di-n-propylessigsaeure
- VALPROIC ACID
- Valproinsaeure
- dipropylacetic acid
- n-DPA
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- Bile salt export pump
- Bile salt export pump (BSEP)
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome P450 2B6
- Cytochrome P450 2J2
- Cytochrome P450 3A
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Frizzled-8
- Glutamate receptor ionotropic, NMDA 1
- Histamine H1 receptor
- Multidrug resistance-associated protein 4
- P2X purinoceptor 4
- Potassium voltage-gated channel subfamily H member 2
- Prion protein
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sodium channel protein type 9 subunit alpha
- Sodium channel protein type I I alpha subunit
- Voltage-gated sodium channel subunit alpha Nav1.4 (Nav1.4)
- 5H-dibenzo[b,f]azepine-5-carboxamide
- CARBAMAZEPINE
- CARBATROL
- CHEMBL108
- DIBENZO[B,F]AZEPINE-5-CARBOXYLIC ACID AMIDE(CARBAMAZEPINE)
- EPITOL
- EQUETRO
- G-32883
- TEGRETOL
- TEGRETOL-XR
- TERIL
- US9138393, Carbamazepine
- US9144538, Carbamazepine
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- Alpha-1A adrenergic receptor
- Beta-1 adrenergic receptor
- Bile salt export pump
- Bile salt export pump (BSEP)
- Cytochrome P450 2D6 (2D6)
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- Histamine H1 receptor
- Monoamine transporter
- Muscarinic acetylcholine receptor M2
- Norepinephrine Monoamine transporters
- Norepinephrine transporter
- Potassium voltage-gated channel subfamily H member 2
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Transporter
- adrenergic Alpha2
- (+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine
- (+/-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine
- (-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine
- (Nomifensine) 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine
- 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine
- 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine (Nomifensine)
- 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine(Nomifensine)
- 2-methyl-4-phenyl-1,2,3,4-tetrahydroisoquinolin-8-amine
- CHEMBL273575
- NOMIFENSINE
- NOMIFENSINE2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine
- Axin-1/Glycogen synthase kinase-3 beta
- Cytochrome P450 2C19
- Cytochrome P450 2C8
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Cytoplasmic tyrosine-protein kinase BMX
- Epidermal growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit alpha
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin receptor
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- MAP kinase-activated protein kinase 2
- MAP kinase-activated protein kinase 3
- Potassium voltage-gated channel subfamily H member 2
- Proto-oncogene tyrosine-protein kinase Src
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase TEC
- Tyrosine-protein kinase TXK
- Tyrosine-protein kinase receptor FLT3
34 IC50
- CHEMBL3263640
- 5-HT3A Serotonin Receptor
- 5-HT5
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2B (5HT2B)
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- D(1A) dopamine receptor
- D(2) dopamine receptor
- HTR1D
- HTR6
- HTR7
- Serotonin (5-HT) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- 2-Me 5-HT
- 2-Methyl-5-hydroxytryptamine
- 2-methyl-5-HT
- 2-methylserotonin
- 3-(2-aminoethyl)-2-methyl-1H-indol-5-ol
- 5-HT,2-Me
- CHEMBL266591
- 3C-like proteinase (3CL-PRO)
- Aldehyde dehydrogenase
- Angiotensin II receptor
- Apelin receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Caspase-1
- Cystic fibrosis transmembrane conductance regulator
- Fatty-acid amide hydrolase 1
- Fructose-1,6-bisphosphatase
- Histone-lysine N-methyltransferase EHMT1
- Lysine-specific demethylase 5A
- Lysyl oxidase
- Lysyl oxidase homolog 2
- Lysyl oxidase homolog 3
- Lysyl oxidase homolog 4
- Monoglyceride lipase
- Multidrug resistance-associated protein 4
- Protein G9a (G9a)
- Replicase polyprotein 1ab
- Transient receptor potential cation channel subfamily A member 1
- perilipin-1
- perilipin-5
- 1,1',1'',1'''-[disulfanediylbis(carbonothioylnitrilo)]tetraethane
- 1,1'-dithiobis(N,N-diethylthioformamide)
- Antabuse (TN)
- CHEMBL964
- DISULFIRAM
- N,N,N',N'-tetraethylthiuram disulfide
- N,N-diethyl[(diethylcarbamothioyl)disulfanyl]carbothioamide (G5)
- bis(diethylthiocarbamoyl) disulfide
- cid_3117
- med.21724, Compound 151
- tetraethylthioperoxydicarbonic diamide
- tetraethylthiuram disulfide
- tetraethylthiuram disulphide
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 2
- D(2) dopamine receptor
- HLA class I histocompatibility antigen A-3
- Histamine H1 receptor
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Norepinephrine transporter
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- 2-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
- CHEMBL621
- TRAZODONE
- Calcium-dependent protein kinase 1 (CDPK1)
- Calmodulin-domain protein kinase 1
- Calmodulin-domain protein kinase 1 (CDPK1)
- Calmodulin-domain protein kinase 1, putative
- Calmodulin/Proto-oncogene tyrosine-protein kinase Src
- Casein kinase I isoform delta
- Cereblon/BCR/ABL
- Cyclin-dependent kinase 2
- Mitogen-activated protein kinase 8
- Phospholipase D (PLD)
- Phospholipase D (PLD_SC)
- Phospholipase D (PLD_sp)
- Phospholipase D2 (PLD2)
- Protein kinase C delta type
- Protein kinase C iota (PKCι)
- Protein kinase C, epsilon
- Protein kinase C, gamma
- Proto-oncogene tyrosine-protein kinase Src
- Serine/threonine-protein kinase D1
- Serine/threonine-protein kinase RIPK2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase CSK
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase LCK
29 IC50
- 1-(1,1-dimethylethyl)-3-(1-naphthalenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
- 1-(tert-butyl)-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine (4)
- 1-NA-PP1
- 1-tert-butyl-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine (4)
- 1-tert-butyl-3-naphthalen-1-yl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
- 4-Amino-1-tert-butyl-3-(1'-naphthyl)pyrazolo[3,4-d]pyrimidine
- CHEMBL264406
- US10544104, Compound 1
- US9765037, Compound 1
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Adrenergic alpha1B
- Alpha-2A adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-3 adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(4) dopamine receptor
- Histamine H1 receptor
- Histamine H2 Receptor
- Histamine H3 receptor
- Mu-type opioid receptor
- Serotonin (5-HT) receptor
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
25 Ki
- (1-(4-fluorophenethyl)piperidin-4-yl)(3-(2-fluoroethoxy)-2-methoxyphenyl)methanol
- (3-(2-Fluoroethoxy)-2-methoxyphenyl)-(1-(2-p-fluorophenylethyl)-piperidine-4-yl)-methanol
- CHEMBL402143
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Adrenergic alpha1B
- Alpha-2A adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-3 adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(4) dopamine receptor
- Histamine H1 receptor
- Histamine H2 Receptor
- Histamine H3 receptor
- Mu-type opioid receptor
- Serotonin (5-HT) receptor
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
24 Ki
- (3-(2-Fluoroethoxy)-2-methoxyphenyl)-(1-(2-p-toluylphenylethyl)-piperidine-4-yl)-methanol
- CHEMBL476839
- Amine oxidase (flavin-containing) A
- Aurora kinase A/B
- Aurora kinase A/Targeting protein for Xklp2
- BRAF/CRAF
- Calmodulin/Proto-oncogene tyrosine-protein kinase Src
- Casein kinase II subunit alpha
- Cyclin-Dependent Kinase 4 (CDK4)
- Cyclin-dependent kinase 2
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Focal adhesion kinase 1/vascular endothelial growth factor receptor 3
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- Mitogen-activated protein kinase kinase kinase 8
- NUAK family SNF1-like kinase 1
- Platelet-derived growth factor receptor beta
- RAC-alpha serine/threonine-protein kinase
- Receptor tyrosine-protein kinase erbB-2
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase PLK4
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
26 IC50
- Alternariol 5-O-Methyl Ether
- CHEMBL483526
- Aurora kinase B
- Cyclin-dependent kinase 2
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 1
- Fibroblast growth factor receptor 2
- Hepatocyte growth factor receptor
- Insulin-like growth factor I receptor
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Protein kinase C alpha type
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAC-alpha serine/threonine-protein kinase
- RAF proto-oncogene serine/threonine-protein kinase
- Receptor protein-tyrosine kinase erbB-4
- Receptor tyrosine-protein kinase erbB-2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
24 IC50
- (S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)-7-(2-methoxyethoxy)quinazolin-6-yl]pyrrolidine-2-carboxamide
- CHEMBL571040
- Aurora kinase B
- Cyclin-dependent kinase 2
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 1
- Fibroblast growth factor receptor 2
- Hepatocyte growth factor receptor
- Insulin-like growth factor I receptor
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Protein kinase C alpha type
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAC-alpha serine/threonine-protein kinase
- RAF proto-oncogene serine/threonine-protein kinase
- Receptor protein-tyrosine kinase erbB-4
- Receptor tyrosine-protein kinase erbB-2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
24 IC50
- (S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylamino)-7-(2-methoxyethoxy)quinazolin-6-yl]pyrrolidine-2-carboxamide
- CHEMBL569880
- Bile salt export pump
- Calcium channel (Type L)
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Carbonic Anhydrase III
- Carbonic Anhydrase VA
- Carbonic Anhydrase VB
- Carbonic Anhydrase XIV
- Carbonic anhydrase 1
- Carbonic anhydrase 12
- Carbonic anhydrase 13 (CA XIII)
- Carbonic anhydrase 15
- Carbonic anhydrase 2
- Carbonic anhydrase 4
- Carbonic anhydrase 6 (CA-VI)
- Carbonic anhydrase 7
- Carbonic anhydrase 9
- Multidrug resistance-associated protein 4
- Potassium voltage-gated channel subfamily H member 2
- Sodium channel protein type 5 subunit alpha
- Sodium channel protein type 9 subunit alpha
- Sodium channel protein type III alpha subunit
- Voltage-gated potassium channel beta subunit Mink/subunit Kv7.1
- Voltage-gated sodium channel subunit alpha Nav1.8
- (2R)-2-acetylamino-N-benzyl-3-methoxypropanamide
- (R)-2-Acetylamino-N-benzyl-3-methoxy-propionamide
- (R)-2-acetamido-N-benzyl-3-methoxypropanamide
- (R)-N-benzyl 2-acetamido-3-methoxypropionamide
- (R)-N-benzyl 2-acetamido-3-methoxypropionamide,
- CHEMBL58323
- Erlosamide
- LACOSAMIDE
- 3-phosphoinositide dependent protein kinase-1
- Cyclin-dependent kinase 1
- Cyclin-dependent kinase 2
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin-like growth factor I receptor
- MAP kinase-activated protein kinase 2
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 8
- Mitogen-activated protein kinase kinase kinase 8
- Mitogen-activated protein kinase kinase kinase kinase 2
- PKC alpha and beta-2
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- Protein kinase C alpha type
- Proto-oncogene tyrosine-protein kinase Src
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 1
- Serine/threonine-protein kinase B-raf
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase PLK1
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase Lck
25 IC50
- CHEMBL1089082
- N-(3-(2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-3-(trifluoromethyl)benzamide
- ALK tyrosine kinase receptor
- Angiopoietin-1 receptor
- CDK2/Cyclin A/Cyclin A1
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 3
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- Lysyl-tRNA synthetase
- Mast/stem cell growth factor receptor Kit
- Platelet-derived growth factor receptor alpha
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAC-alpha serine/threonine-protein kinase
- Receptor tyrosine-protein kinase erbB-2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase HCK
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase ZAP-70
- Vascular endothelial growth factor receptor 2
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
25 IC50
- CHEMBL1085511
- isobutyl4-(7-amino-3-(4-(4-methylpiperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-6-yl)phenylcarbamate
- Aurora kinase B
- CaM kinase IV
- Casein kinase I isoform delta
- Cyclin-dependent kinase 2
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Hepatocyte growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- Mitogen-activated protein kinase 1
- Protein kinase C alpha type
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase alpha-3
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase Nek2
- Serine/threonine-protein kinase PLK3
- Testis-specific serine/threonine-protein kinase 2
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 2
27 IC50
- 2-(ethyl((5-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-ylamino)isothiazol-3-yl)methyl)amino)-2-methylpropan-1-ol
- 2-{ethyl[(5-{[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-ol
- CHEMBL1232515
- CHEMBL1650533
- Cytochrome P450 1A
- Cytochrome P450 2C19
- Cytochrome P450 2C9
- Cytochrome P450 2D6 (2D6)
- Cytochrome P450 3A
- Diacylglycerol O-acyltransferase 1 (DGAT1)
- Fibroblast growth factor receptor 1
- Insulin-like growth factor I receptor
- MAP kinase-activated protein kinase 2
- Mitogen-activated protein kinase 14
- Non-receptor tyrosine-protein kinase TYK2
- PKC alpha and beta-2
- Potassium voltage-gated channel subfamily H member 2
- Protein kinase C (PKC)
- Protein kinase C alpha type
- Protein kinase C delta type
- Serine/threonine-protein kinase PLK1
- Signal transducer and activator of transcription 3
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
- Vascular endothelial growth factor receptor 2
24 IC50
- 5-amino-1-(2-fluorophenyl)-N-(5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl)-1H-pyrazole-4-carboxamide
- CHEMBL1290746
- Aurora kinase B
- CaM kinase IV
- Casein kinase I isoform delta
- Cyclin-dependent kinase 2
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Hepatocyte growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- Mitogen-activated protein kinase 1
- Protein kinase C alpha type
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase alpha-3
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase Nek2
- Serine/threonine-protein kinase PLK3
- Testis-specific serine/threonine-protein kinase 2
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 2
48 IC50
- CHEMBL1650545
- CHEMBL1650551
- N-[3-[(3,3-Difluoro-1-pyrrolidinyl)methyl]-5-isothiazolyl]-6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amine Hydrochloride
- 17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3)
- Aldo-keto reductase family 1 member C1
- Aldo-keto reductase family 1 member C2
- Aldo-keto reductase family 1 member C4 (AK1C4)
- Aldo-keto-reductase family 1 member C3
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Caspase-1
- Caspase-3
- Caspase-4
- Caspase-5
- Caspase-9
- Cyclooxygenase
- Cyclooxygenase-1 (COX-1)
- Cytochrome P450 2J2
- Dihydrofolate reductase
- Multidrug resistance-associated protein 4
- Prostaglandin E synthase/G/H synthase 2
- Prostaglandin G/H synthase (Cyclooxygenase-2)
- Prostaglandin G/H synthase (cyclooxygenase)
- Prostaglandin-H2 D-isomerase
- Seed lipoxygenase-1
- Solute carrier family 22 member 6
- (2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid
- (S)-2-(6-Methoxy-naphthalen-2-yl)-propionic acid
- (S)-2-(6-methoxynaphthalen-2-yl)propanoic acid
- (S)-naproxen
- 2-(6-Methoxy-naphthalen-2-yl)-propionic acid
- 2-(6-Methoxy-naphthalen-2-yl)-propionic acid(naproxen)
- 2-(6-methoxy-2-naphthyl)propanoic acid
- 2-(6-methoxynaphthalen-2-yl)propanoic acid
- Aleve
- Anaprox
- CHEMBL154
- Ec-naprosyn
- Equiproxen
- Naprelan
- Naprosyn
- Naproxen
- Naproxen2-(6-Methoxy-naphthalen-2-yl)-propionic acid
- RS-3540
- S-NAPROXEN
- naproxene
- Adenylate kinase 1
- Adenylate kinase 2
- Glycerol kinase
- Heat shock protein 75 kDa, mitochondrial
- Heat shock protein 90 beta
- Ketopantoate reductase
- MAP kinase-activated protein kinase 2
- Mitogen-activated protein kinase kinase kinase 7
- P2X purinoceptor 1
- P2X purinoceptor 3
- P2X purinoceptor 4
- P2X purinoceptor 5
- P2X purinoceptor 6
- P2X purinoceptor 7
- P2Y purinoceptor 1
- Purinergic receptor P2Y1
- Purinergic receptor P2Y11
- Purinergic receptor P2Y12
- Purinergic receptor P2Y2
- Purinergic, P2X2
- Pyrimidinergic receptor P2Y4
- Pyrimidinergic receptor P2Y6
- Serine/threonine protein phosphatase 2A, 56 kDa regulatory subunit, alpha isoform
- Tyrosine-protein kinase JAK2
- ADENOSINE TRIPHOSPHATE
- ATP
- Adrenaline alpha1
- Adrenaline alpha2
- Adrenergic Alpha
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cystic fibrosis transmembrane conductance regulator
- Cytochrome P450 2D1
- Cytochrome P450 2D18
- Cytochrome P450 2D2
- Cytochrome P450 2D3
- Cytochrome P450 2D6
- Cytochrome P450 2D6 (2D6)
- Histidine-rich protein
- Multidrug resistance protein 1/Multidrug resistance associated protein 1
- Multidrug resistance-associated protein 4
- P-glycoprotein 1
- Serum albumin
- Sodium channel protein type I I alpha subunit
- Solute carrier family 22 member 1
- Solute carrier family 22 member 2
- Solute carrier organic anion transporter family member 1A1
- Solute carrier organic anion transporter family member 1A4
- Twik-RElated Potassium (K+) channel 1 (TREK1)
- QUININE
- Quinamm
- Quinsan
- cid_3034034
- 10 kDa chaperonin
- 60 kDa heat shock protein, mitochondrial
- Arylacetamide deacetylase
- Bile salt export pump
- Bile salt export pump (BSEP)
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome P450 2B6
- DNA gyrase subunit B
- Enoyl-ACP Reductase (InhA)
- Glutathione transferase omega 1
- Multidrug resistance-associated protein 4
- NH(3)-dependent NAD(+) synthetase
- Nuclear receptor subfamily 1 group I member 2
- RNA polymerase beta subunit (EC 2.7.7.6)
- Serum albumin
- Solute carrier organic anion transporter family member 1A1
- Solute carrier organic anion transporter family member 1A2
- Solute carrier organic anion transporter family member 1A4
- Solute carrier organic anion transporter family member 1B1 (OATP1B1)
- Solute carrier organic anion transporter family member 1B3 (OATP1B3)
- Solute carrier organic anion transporter family member 2B1
- Sterol 14α-demethylase (CYP51)
- Thiosulfate sulfurtransferase
- BA-41166E
- L-5103
- RIFAMPIN
- Rifadin
- Rifampicin
- ALK tyrosine kinase receptor
- Cytoplasmic tyrosine-protein kinase BMX
- Ephrin type-A receptor 3
- Ephrin type-B receptor 2
- Fibroblast growth factor receptor
- High affinity nerve growth factor receptor
- Insulin receptor
- Insulin-like growth factor 1 receptor
- JNK1/JNK2
- Macrophage colony-stimulating factor 1 receptor (c-Fms)
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- NT-3 growth factor receptor
- Neuronal proto-oncogene tyrosine-protein kinase Src
- Platelet-derived growth factor receptor beta
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Receptor-type tyrosine-protein kinase FLT3
- TPR/MET fusion protein
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor Tie-1
- Vascular endothelial growth factor receptor 1
25 IC50
- CHEMBL2037224
- ALK tyrosine kinase receptor
- Cytoplasmic tyrosine-protein kinase BMX
- Ephrin type-A receptor 3
- Ephrin type-B receptor 2
- Fibroblast growth factor receptor
- High affinity nerve growth factor receptor
- Insulin receptor
- Insulin-like growth factor 1 receptor
- JNK1/JNK2
- Macrophage colony-stimulating factor 1 receptor (c-Fms)
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- NT-3 growth factor receptor
- Neuronal proto-oncogene tyrosine-protein kinase Src
- Platelet-derived growth factor receptor beta
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Receptor-type tyrosine-protein kinase FLT3
- TPR/MET fusion protein
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor Tie-1
- Vascular endothelial growth factor receptor 1
25 IC50
- CHEMBL2037208
- ALK tyrosine kinase receptor
- BDNF/NT-3 growth factors receptor
- Cytoplasmic tyrosine-protein kinase BMX
- Ephrin type-A receptor 3
- Ephrin type-B receptor 2
- Fibroblast growth factor receptor
- High affinity nerve growth factor receptor
- Insulin receptor
- Insulin-like growth factor 1 receptor
- JNK1/JNK2
- Macrophage colony-stimulating factor 1 receptor (c-Fms)
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Neuronal proto-oncogene tyrosine-protein kinase Src
- Platelet-derived growth factor receptor beta
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Receptor-type tyrosine-protein kinase FLT3
- TPR/MET fusion protein
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor Tie-1
- Vascular endothelial growth factor receptor 1
26 IC50
- CHEMBL2037226
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Delta-type opioid receptor
- Histamine H1 receptor
- Histamine H2 receptor
- Histamine H3 receptor
- Histamine H4 receptor
- Kappa-type opioid receptor
- Mu-type opioid receptor
- Nitric Oxide Synthase, endothelial
- Nitric Oxide Synthase, inducible
- Nitric oxide synthase, brain
- Nitric oxide synthase, endothelial
- Nitric oxide synthase, inducible
- Nitric-oxide synthase, brain
- Nitric-oxide synthase, endothelial
- Nociceptin receptor
- Serotonin (5-HT) receptor
47 Ki
- CHEMBL3126204
- US9212144, 15 (Ex. 17)
- Aurora kinase A/Targeting protein for Xklp2
- Aurora kinase B
- Axin-1/Glycogen synthase kinase-3 beta
- CaM kinase IV
- Casein kinase I isoform delta
- Cyclin-dependent kinase 2
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Hepatocyte growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin-like growth factor I receptor
- Mitogen-activated protein kinase 1
- PKC alpha and beta-2
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase alpha-1/alpha-3
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase NEK2
- Serine/threonine-protein kinase PLK3
- Testis-specific serine/threonine-protein kinase 2
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase receptor FLT3
- CHEMBL4228240
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2C adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- HTR1D
- HTR2C
- Histamine H1 receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Serotonin 1B/1D receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Voltage-gated sodium channel subunit alpha Nav1.8
- adrenergic Alpha2
27 Ki
- CAS_6438382
- NSC_6438382
- SR 46349B
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-2 adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- HTR2C
- Histamine H1 receptor
- Monoamine transporters; Norepininephrine & dopamine
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Norepinephrine Monoamine transporters
- Norepinephrine transporter
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Transporter
- adrenergic Alpha2
- CHEMBL284994
- CP-52003
- SERTRALINE
- [4-(3,4-Dichloro-phenyl)-1,2,3,4-tetrahydro-naphthalen-1-yl]-methyl-amine
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Histamine H1 receptor
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Norepinephrine transporter
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- adrenergic Alpha2
- CAS_23047-25-8
- Lofepramine
- NSC_3947
- US8629135, SW-06