Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- 5-HT1
- 5-HT3A Serotonin Receptor
- 5-HT5
- 5-HT5B
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2B (5HT2B)
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- 5-hydroxytryptamine receptor 7 (5HT7)
- ADRA1A
- ADRA1B
- Adrenergic alpha1B
- Adrenergic receptor
- Adrenergic receptor alpha-2
- Alpha adrenergic receptor 1A and 1B
- Alpha adrenergic receptor 1A and 1D
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-1D adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-casein
- Bile salt export pump
- Cerebral cortex alpha adrenergic receptor
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- DRD1
- DRD2
- Dopamine D1 receptor
- Dopamine D1B
- Dopamine receptor
- HLA class I histocompatibility antigen A-3
- HTR1D
- HTR2B
- HTR2C
- HTR6
- HTR7
- Histamine H1 receptor
- Muscarinic acetylcholine receptor
- Muscarinic acetylcholine receptor M2
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sigma non-opioid intracellular receptor 1
- Sodium channel protein type I I alpha subunit
- Sodium-dependent serotonin transporter
- Sphingosine 1-phosphate receptor 3
- Vesicular acetylcholine transporter
- adrenergic Alpha1
- adrenergic Alpha2
- 8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
- 8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
- 8-[4-(4-fluorophenyl)-4-oxobutyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
- CHEMBL267930
- MLS000028615
- SMR000058674
- SPIPERONE
- Spiroperidol
- US9359372, Spiperone
- [3H]-Spiroperidol
- cid_5265
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- ADENOSINE A2
- ADRA2B
- Adenosine receptor A1
- Adenosine transporter
- Adenylate cyclase Forskolin
- Alpha adrenergic receptor 1A and 1B
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Calcium channel (Type T,L)
- Cholecystokinin receptor
- Cytochrome P450 2D6 (2D6)
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Ecto-5'-nucleotidase (e5'NT)
- GRIA3
- Gamma-aminobutyric acid receptor subunit alpha-1
- Gamma-aminobutyric acid type B receptor subunit 1
- Glutamate receptor ionotropic, NMDA 1
- Glutamate receptor ionotropic, kainate 1
- Glycine receptor subunit alpha-1
- Glycine, non-strychnine
- HTR4
- Histamine H1 receptor
- Histamine H2 receptor
- Inositol Triphosphate
- Kappa-type opioid receptor
- Melatonin receptor
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Neurokinin 1 receptor
- Neurokinin 2 receptor
- Neurokinin 3 receptor
- Neuropeptide Y receptor type 1
- Nitric-oxide synthase, brain
- Nociceptin receptor
- Norepinephrine transporter
- Opioid receptors; mu & delta
- Potassium Channel
- Protein kinase C
- Renal Outer Medullary Potassium (ROMK)
- SOMATOSTATIN
- Sigma non-opioid intracellular receptor 1
- Sodium (Site 1)
- Sodium (Site 2)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Voltage-dependent N-type calcium channel subunit alpha-1B
- adrenergic Alpha2
- alpha-1 Nicotinic AChR
- (R)-N-methyl-3-phenyl-3-(o-tolyloxy)propan-1-amine
- ATOMOXETINE
- CHEMBL641
- Methyl-((R)-3-phenyl-3-o-tolyloxy-propyl)-amine
- Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine
- Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxetine)
- Strattera
- Tomoxetine
- 1,3-beta-glucan synthase component GLS2
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Adrenergic alpha1B
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Delta-type opioid receptor
- Dopamine D1B
- Dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- Gamma-aminobutyric acid type B receptor subunit 1
- Glutamate receptor ionotropic, NMDA 1
- HRH3
- HTR6
- Histamine H1 receptor
- Histamine H2 Receptor
- Histamine H4 receptor
- Histone H1
- Kappa-type opioid receptor
- Mu-type opioid receptor
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M1 and M3
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- P-glycoprotein 1
- Potassium voltage-gated channel subfamily H member 2
- Prostaglandin E2 receptor
- Prostaglandin E2 receptor EP4 subtype
- Protein kinase C alpha type
- Protein kinase C, gamma
- Serotonin (5-HT) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Solute carrier family 22 member 2
- 7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one
- ARIPIPRAZOLE
- CHEMBL1112
- US10174011, aripiprazole
- US10752588, Compound Aripiprazole
- US9018213, aripprazole
- US9156822, Aripiprazole
- ALK tyrosine kinase receptor
- Activin receptor type-1
- Aurora kinase A/Targeting protein for Xklp2
- Aurora kinase B
- Axin-1/Glycogen synthase kinase-3 beta
- BDNF/NT-3 growth factors receptor
- CAMK2A
- CaM kinase I delta
- Casein kinase I isoform alpha
- Cyclin-dependent kinase 7
- Cyclin-dependent kinase 8
- Cyclin-dependent kinase 9
- Death-associated protein kinase 3
- Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
- Dual specificity mitogen-activated protein kinase kinase; MEK1/2
- Dual specificity protein kinase CLK2
- Dual specificity protein kinase TTK
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Fibroblast growth factor receptor 1
- Focal adhesion kinase 1
- G protein-coupled receptor kinase 5
- Glycogen synthase kinase-3
- Hepatocyte growth factor receptor
- Hepatocyte growth factor-like protein
- High affinity nerve growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon
- Insulin receptor
- Insulin-like growth factor I receptor
- Leukocyte tyrosine kinase receptor
- Macrophage colony-stimulating factor 1 receptor (CSF1R)
- Mitogen-activated protein kinase 8
- Mitogen-activated protein kinase 9
- Mitogen-activated protein kinase kinase kinase kinase 2
- Mitogen-activated protein kinase kinase kinase kinase 4
- NT-3 growth factor receptor
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Protein kinase C theta type
- Protein kinase C, PKC; classical/novel
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase alpha-1/alpha-3
- Serine/threonine-protein kinase NEK2
- Serine/threonine-protein kinase PAK 4
- Serine/threonine-protein kinase TAO2
- Serine/threonine-protein kinase TBK1
- Serine/threonine-protein kinase WEE1
- Serine/threonine-protein kinase pim-1
- Tyrosine kinase non-receptor protein 2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase receptor TYRO3
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- CHEMBL4078893
- ALK tyrosine kinase receptor
- Activin receptor type-1
- Aurora kinase A/Targeting protein for Xklp2
- Aurora kinase B
- Axin-1/Glycogen synthase kinase-3 beta
- BDNF/NT-3 growth factors receptor
- CAMK2A
- CaM kinase I delta
- Casein kinase I isoform alpha
- Cyclin-dependent kinase 7
- Cyclin-dependent kinase 8
- Cyclin-dependent kinase 9
- Death-associated protein kinase 3
- Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
- Dual specificity mitogen-activated protein kinase kinase; MEK1/2
- Dual specificity protein kinase CLK2
- Dual specificity protein kinase TTK
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Fibroblast growth factor receptor 1
- Focal adhesion kinase 1
- G protein-coupled receptor kinase 5
- Glycogen synthase kinase-3
- Hepatocyte growth factor receptor
- Hepatocyte growth factor-like protein
- High affinity nerve growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon
- Insulin receptor
- Insulin-like growth factor I receptor
- Leukocyte tyrosine kinase receptor
- Macrophage colony-stimulating factor 1 receptor (CSF1R)
- Mitogen-activated protein kinase 8
- Mitogen-activated protein kinase 9
- Mitogen-activated protein kinase kinase kinase kinase 2
- Mitogen-activated protein kinase kinase kinase kinase 4
- NT-3 growth factor receptor
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Protein kinase C theta type
- Protein kinase C, PKC; classical/novel
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Serine/threonine-protein kinase 16
- Serine/threonine-protein kinase NEK2
- Serine/threonine-protein kinase PAK 4
- Serine/threonine-protein kinase TAO2
- Serine/threonine-protein kinase TBK1
- Serine/threonine-protein kinase WEE1
- Serine/threonine-protein kinase pim-1
- Tyrosine kinase non-receptor protein 2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase receptor TYRO3
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- CHEMBL4062803