Compile Data Set for Download or QSAR
Report error Found 132 Enz. Inhib. hit(s) with Target = 'UDP-N-acetylmuramoylalanine--D-glutamate ligase'
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119097(MurD inhibitor (compound 36))
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119123(MurD/E/F inhibitor (compound 69))
Affinity DataIC50: 2.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM26455(MurD inhibitor (compound 40) | (2R)-2-({6-[(4-cyan...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to 6x His-tagged and 15N/13C-labeled Escherichia coli MurD ligase measured at NMR signal 9 by 1H/13C-HSQC 2D NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119104(MurD inhibitor (compound 46))
Affinity DataIC50: 3.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM26455(MurD inhibitor (compound 40) | (2R)-2-({6-[(4-cyan...)
Affinity DataKd:  5.50E+3nMAssay Description:Binding affinity to 6x His-tagged and 15N/13C-labeled Escherichia coli MurD ligase measured at NMR signal 56 by 1H/13C-HSQC 2D NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM119107(MurD/E inhibitor (compound 49))
Affinity DataIC50: 6.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM26455(MurD inhibitor (compound 40) | (2R)-2-({6-[(4-cyan...)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to 6x His-tagged and 15N/13C-labeled Escherichia coli MurD ligase measured at NMR signal 13 by 1H/13C-HSQC 2D NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119107(MurD/E inhibitor (compound 49))
Affinity DataIC50: 8.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119100(MurD inhibitor (compound 42))
Affinity DataIC50: 8.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119105(MurD inhibitor (compound 47))
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475587(CHEMBL426651)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475586(CHEMBL198030)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475591(CHEMBL382328)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM119122(MurA/B/C/D/E inhibitor (compound 67))
Affinity DataIC50: 1.30E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475590(CHEMBL370421)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475579(CHEMBL382202)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM85276(MurC/D/E/F inhibitor (compound 68) | HEA derivativ...)
Affinity DataIC50: 1.80E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475601(CHEMBL199812)
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475599(CHEMBL200097)
Affinity DataIC50: 2.05E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.10E+4nMAssay Description:Competitive inhibition of Escherichia coli MurD using D-Glu substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475603(CHEMBL199320)
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.90E+4nMAssay Description:Partial non-competitive inhibition of Escherichia coli MurD using UMA substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119086(MurD inhibitor (compound 35) | MurC/D inhibitor (c...)
Affinity DataIC50: 3.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119086(MurD inhibitor (compound 35) | MurC/D inhibitor (c...)
Affinity DataIC50: 3.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221037(CHEMBL87262)
Affinity DataIC50: 3.02E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221022(CHEMBL86525)
Affinity DataIC50: 3.28E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475582(CHEMBL199511)
Affinity DataIC50: 3.35E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221032(CHEMBL86526)
Affinity DataIC50: 3.45E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475607(CHEMBL199629)
Affinity DataIC50: 3.47E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221030(CHEMBL313078)
Affinity DataIC50: 3.60E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  3.90E+4nMAssay Description:Partial un-competitive inhibition of Escherichia coli MurD using ATP substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221020(CHEMBL87126)
Affinity DataIC50: 4.19E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119122(MurA/B/C/D/E inhibitor (compound 67))
Affinity DataIC50: 4.40E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119106(MurD inhibitor (compound 48))
Affinity DataIC50: 4.50E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM119103(MurD inhibitor (compound 45))
Affinity DataIC50: 4.50E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2014
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221027(CHEMBL327438)
Affinity DataIC50: 4.52E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221018(CHEMBL85772)
Affinity DataIC50: 4.74E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221038(CHEMBL87521)
Affinity DataIC50: 4.87E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475596(CHEMBL200015)
Affinity DataIC50: 4.88E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221023(CHEMBL84684)
Affinity DataIC50: 4.93E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221033(CHEMBL420601)
Affinity DataIC50: 4.97E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475600(CHEMBL381006)
Affinity DataIC50: 5.32E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50475597(CHEMBL380752)
Affinity DataIC50: 5.32E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475593(CHEMBL199553)
Affinity DataIC50: 5.86E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475595(CHEMBL199757)
Affinity DataIC50: 6.12E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus)
University of Ljubljana

LigandPNGBDBM50221019(CHEMBL87584)
Affinity DataIC50: 6.37E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2018
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475602(CHEMBL199929)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475584(CHEMBL197817)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
University of Ljubljana

LigandPNGBDBM50475606(CHEMBL199580)
Affinity DataIC50: 6.53E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 132 total ) | Next | Last >>
Jump to: