Compile Data Set for Download or QSAR
Report error Found 354 Enz. Inhib. hit(s) with all data for entry = 10809
TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510491BDBM510491((5S)-N-(2,4- clichlorebenzyl)-5- fluoro-8-((2- hyd...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510492BDBM510492((5R,8S)-N-(2-chloro-3- (trifluoromethyl)benzyl)- 5...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510477BDBM510477((5S,8S)-N- (2-chloro-4- fluorobenzyl)- 5-fluoro-8-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510478BDBM510478((5S,8S)-N- (2-chloro-4- (trifluoromethyl) benzyl)-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 570856BDBM570856((5S,8S)-N-(2,4-dichloro- 6-fluorobenzyl)-5-fluoro-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510476BDBM510476((5S,8S)-N-(2,3- dichlorobenzyl)- 5-fluoro-8- hydro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510479BDBM510479((5S,8S)-5-fluoro-8- methoxy-N-(2,3,4- trifluorobe...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510480BDBM510480((5S,8S)-N- (4-chloro-2- fluorobenzyl)- 5-fluoro-8-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510485BDBM510485((5S,8S)-5-fluoro-8-(2- hydroxyethoxy)-N- (2.3.4-tr...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510486BDBM510486((5S,8S)-N-(4-chloro-2- fluorobenzyl)-5-fluoro-8- (...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510483BDBM510483((5S,8S)-N-(2,4-dichloro- 6- (hydroxymethyl)benzyl)...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510484BDBM510484((5S,8S)-N-(2-chloro-4- fluorobenzyl)-5-fluoro-8- (...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510489BDBM510489((5S,8S) N-(2,4-dichlorobenzyl)-8-(2,3-dihydroxypro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510490BDBM510490((5S)-N-(2,4- dichlorobenzyl)-5- fluoro-8- (methyls...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510033BDBM510033(N-(2,4-dichloro-6-methyl- benzyl)-8-oxo-5,6,7,8- t...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510052BDBM510052(N-(2-chloro-3-(trifluoro methyl)benzyl)-8-oxo-5, 6...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510097BDBM510097(N-(2,4-dichloro-6-methyl- benzyl)-8-hydroxy-5,6, 7...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510061BDBM510061(N-(2,4-dichloro-6-(hydroxy- methyl)benzyl)-8-oxo- ...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510149BDBM510149(N-(2,4-dichloro-6-(hydroxy- methyl)benzyl)-8-hydro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510150BDBM510150(N-(2,4-dichloro-6-(methoxy- methyl)benzyl)-8-hydro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510147BDBM510147(N-(2-chloro-3-(trifluoro methyl)benzyl)-8-hydroxy-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510148BDBM510148(N-(2,3-dichlorobenzyl)- 8-hydroxy-5,6,7,8-tetra hy...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510153BDBM510153(N-(2-chloro-3-(trifluoromethyl)benzyl)- 5-fluoro-8...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510154BDBM510154(N-(2,4-dichloro-6-(hydroxymethyl) benzyl)-5-fluoro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510151BDBM510151(N-(2,4-dichloro-6-methyl- benzyl)-7-methylene- 6,7...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510152BDBM510152(N-(2,4-dichloro-6-methylbenzyl)-5- fluoro-8-oxo-5,...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510173BDBM510173(N-(2,4-dichloro-6-methylbenzyl)-8-hy- droxy-8-(hyd...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510174BDBM510174(N-(2,4-dichloro-6-methylbenzyl)-5- fluoro-8-hydrox...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510172BDBM510172((2-amino-2-oxoethyl)-N- (2-chloro-3-(trifluoro- me...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510177BDBM510177(N-(2,4-dichlorobenzyl)-5-fluoro-8-hy- droxy-8-(hyd...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510175BDBM510175(N-(2-chloro-3-(trifluoromethyl)benzyl)- 5-fluoro-8...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510176BDBM510176(N-(2,3-dichlorobenzyl)-5-fluoro-8-hy- droxy-8-(hyd...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510181BDBM510181((5S*,8S*)-N-(2,4- dichlorobenzyl)- 5-fluoro-8-hydr...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510182BDBM510182((5S*,8S*)-N-(2- chloro-4-fluoro- benzyl)-5-fluoro-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 570506BDBM570506(N-(2,4-dichloro-6-meth- ylbenzyl)-5-fluoro-8-hy- d...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510180BDBM510180(N-(2-chloro-3-(tri- fluoromethyl)benzyl)- 5-fluoro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510185BDBM510185(8-(aminomethyl)- N-(2,4-dichloro-6- methylbenzyl)-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510186BDBM510186(N-(2,4-dichloro-6- methylbenzyl)- 5-fluoro-8- hydr...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510183BDBM510183(8-(aminomethyl)-N- (2,4-dichloro-6-meth- ylbenzyl)...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510184BDBM510184(N-(2,4-dichloro-6- methylbenzyl)-8- hydroxy-8-((me...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510158BDBM510158(N-(2,4-dichloro-6-methyl- benzyl)-5-fluoro-8-hydro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510156BDBM510156(N-(2,4-dichloro-6-methylbenzyl)-7-oxo- 6,7-dihydro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510161BDBM510161(N-(2,3-dichlorobenzyl)-5- fluoro-8-hydroxy-5,6,7,8...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510162BDBM510162(N-(2,4-dichlorobenzyl)-5- fluoro-8-hydroxy-5,6,7,8...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510159BDBM510159(N-(2-chloro-3-(trifluoro- methyl)benzyl)-5-fluoro-...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510160BDBM510160(N-(2,4-dichloro-6-(hydroxy methyl)benzyl)-5-fluoro...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510166BDBM510166(N-(2,4-dichloro-6-methyl- benzyl)-7-hydroxy-6,7- d...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510163BDBM510163(N-(2,4-dichloro-6-(methoxy- methyl)benzyl)-5-fluor...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510164BDBM510164(N-(2,4-dichloro-6-methyl- benzyl)-5,8-dihydroxy-5,...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Raqualia Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 510169BDBM510169(N-(2,4-dichlorobenzyl)-5- fluoro-7-hydroxy-6,7-dih...)
Affinity DataIC50: 50nMAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

Displayed 1 to 50 (of 354 total ) | Next | Last >>
Jump to: