TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of human LSD1/CoRESTMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of human LSD1/CoRESTMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of human LSD1/CoRESTMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
Affinity DataKi: 640nMAssay Description:Inhibition of human LSD1/CoRESTMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 950nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of human LSD1 using K4me2 peptide as substrate measured after 10 mins by peroxidase-coupled reaction assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 760nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH] FabI(Escherichia coli)
Meiji Seika Kaisha
Curated by ChEMBL
Meiji Seika Kaisha
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of Escherichia coli enoyl-ACP reductase FabIMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Streptococcus pneumoniae KU197 FabKMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Streptococcus pneumoniae FabKMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Streptococcus pneumoniae enoyl-ACP reductase FabKMore data for this Ligand-Target Pair